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ABOUT US
Shanghai angti biotechnology co., LTD., founded in 2014, is a research and development focus on pharmaceutical intermediates and apis and process optimization of the production company. Company is located in zhangjiang high-tech park Shanghai pudong, the company's technology and research and development strength, is a high-tech enterprise of be worthy of the name.
Company since its inception, always adhere to the talent for this, the principle of sincerity, make the enterprise in the fierce market competition always remain competitive, to reach the company fast and steady development. Company personnel reasonable structure, has doctor, master's, bachelor's degree high, intermediate technical titles, such as multi-level employees. Provides technical support for the development of the company, the abundant technical strength, excellent product quality will become your most reliable long-term partner.

Products
Biluding block
   tert-ButylMalononitrile 
   2,3-Dimethoxybenzyl alcohol 
   2,6-Dimethyl-3,5-heptanedione 
   3-Methylpyridin-2-ol 
   2-Hydroxythioanisole 
   2-(Methylthio)aniline 
   5-Ethyl-3-hydroxy-4-methyl-2(5H)-furanone 
   Cyclopentaneacetaldehyde 
   2-Cyclopentylethanol 
   3H-benzo[c][1,2]dithiol-3-one 
   (2,6,6-Trimethyl-2-hydroxycyclohexylidene)acetic acid lactone 
   6,10-Dimethyl-5,9-undecadien-2-one 
   3-amino-3-methyl-1-(1-pyrrolidinyl)-1-Butanone 
   2-hydrazinyl-1-methyl-1H-benzo[d]imidazole 
   1,3-Dibenzylurea 
   1-(6-bromo-1H-pyrrolo[3,2-c]pyridin-1-yl)ethanone 
   tert-Butyl 6-bromo-1H-pyrrolo[3,2-c]pyridine-1-carboxylate 
   3-Chloro-6-(pyridin-2-ylmethyl)pyridazine 
   (3R,4S)-Tetrahydrofuran-3,4-diamine dihydrochloride  
   硫坎酮 
   5,6-dimethylfuro[2,3-d]pyrimidin-4(3H)-one 
   (1-benzylpiperidin-4-yl)methanamine hydrochloride 
   2,6-Dibromotoluene 
   1H-Indole-4-carbaldehyde 
   4-Cyanoindole 
   3-Bromo-2-methylphenol 
   4-Fluorostyrene 
   2-Fluorostyrene 
   3-Fluorostyrene 
   2-Bromostyrene 
   3-Bromostyrene 
   4-Bromostyrene 
   3-Chlorostyrene 
   2-Chlorostyrene 
   4-Chlorostyrene 
   5-AMino-2-naphthol 
   7-IsoquinolinaMine, 1-chloro-3-(3-Methoxyphenyl)-N,N-diMethyl- 
   (3-fluoro-2-(trifluoromethyl)phenyl)boronic acid 
   (2-bromo-3-fluorophenyl)boronic acid 
   3-Fluoro-4-trifluoromethylphenylboronic acid 
   5-Chloro-2-(trifluoromethoxy)phenylboronicacid 
   (5-Chloro-2-fluorophenyl)hydrazine 
   6-bromo-8-methoxyquinoline 
   4-Chloro-7-hydroxyquinoline 
   7-AMinoquinoline 
   3-bromocyclobutanone 
   6-Bromo-2-chloronicotinic acid 
   2,2-dimethylOxazolidine 
   5-Fluoro-2-(trifluoroMethyl)pyridine 
   4-Oxocyclohexanecarboxylic acid 
   1-Phenylpiperidin-4-one 
   3,3,5,5-tetramethylmorpholine 
   4-BroMobenzofuran 
   5-Chlorobenzofuran 
   2,5-dibromofuran 
   2,4-DICHLORO-6-FLUOROPYRIMIDINE 
   2-Chloroquinazoline 
   3-bromo-1H-indole 
   8-hydroxy-3,4-dihydronaphthalen-1(2H)-one 
   4-aminocyclohexanone 
   4-chloro-6,7-dimethoxyquinazolin-2-amine 
   5-chloro-2-nitrobenzoic acid 
   4,6-dichloroquinoline 
   5-chloro-2-(trifluoromethyl)aniline 
   6-chloroindoline 
   4,5-dichloropicolinic acid 
   2-methylnicotinonitrile 
   5-bromo-2-chlorobenzo[d]thiazole 
   4-nitropyridin-3-ol 
   2,2-difluoro-1,3-dimethylimidazolidine 
   4-bromo-3-fluoro-2-methylpyridine 
   2-methyl-2H-tetrazole-5-thiol 
   3-oxo-1,3-dihydroisobenzofuran-5-carbonitrile 
   6-Hydroxy-4-methyl-2H-chromen-2-one 
   2-methylthiazol-5-amine 
   4-nitroisophthalonitrile 
   3-amino-4-nitrobenzoic acid 
   methyl 4-bromo-6-chloronicotinate 
   methyl 2-chloro-5-ethynylnicotinate 
   N-(4-(1-aminoethyl)pyridin-2-yl)propionamide 
   2-(cyclopropylmethoxy)pyridine-4-carbothioamide 
   2-amino-3-(2,4-dichlorophenyl)propanenitrile 
   2-(cyclopropylmethoxy)isonicotinonitrile 
   2-(bromomethyl)-3,5-dichloropyridine 
   N-(4-(aminomethyl)-6-methylpyridin-2-yl)propionamide 
   5-iodopyrimidin-4-amine 
   4-bromo-3-(trifluoromethyl)pyridine 
   4-methoxypyridin-2-amine 
   oxazolidine 
   2-fluorocyclohexanone 
   2-chloro-4-methoxy-7H-pyrrolo[3,4-d]pyrimidine 
   3-Boc-1,2,3-oxathiazolidine 2,2-dioxide 
   5-amino-2-nitrobenzoic acid 
   4H-pyran-4-one 
   3-chloro-4-(trifluoromethyl)aniline 
   2-Cyano-6-isopropylpyridine 
   3-(bromomethyl)oxetane 
   oxetan-3-ylmethanol 
   4-hydroxypyrazole 
   4-ethoxy-1H-pyrazole 
   4-methoxy-1H-pyrazole 
   4-ethyl-1H-pyrazole 
   4-propan-2-yl-1H-pyrazole 
   4-cyclopropyl-1H-pyrazole hydrochloride 
   5-ethyl-1H-pyrazole-3-carboxylic acid 
   5-bromo-1-methylpyrazole-3-carboxylic acid 
   5-bromo-1-methylpyrazol-3-amine 
   methyl 5-bromo-1H-pyrazole-3-carboxylate 
   5-BroMo-1H-pyrazole-3-carboxylic acid 
   5-bromo-1H-pyrazole-3-carbaldehyde 
   2-amino-4-methyl-picolinic acid methyl ester 
   6-amino-3-methyl-pyridine-2-carboxylic acid methyl ester 
   3-(bromomethyl)-1,1-difluorocyclobutane 
   tert-butyl 6-amino-2-azaspiro[3.4]octane-2-carboxylate 
   tert-butyl 7-amino-2-azaspiro[4.4]nonane-2-carboxylate 
   tert-butyl (2-azaspiro[4.4]nonan-7-yl)carbamate 
   tert-butyl (2-azaspiro[3.4]octan-6-yl)carbamate 
   2-Oxo-pyrrolidine-3-carboxylic acid 
   ethyl 2-oxopyrrolidine-3-carboxylate 
   1-piperidin-4-ylazepane 
   Piperazine,1-(1-methylethyl)-4-phenyl-  
   4-(oxan-4-yl)aniline 
   4-phenyloxane 
   1-Piperidin-4-yl-4-propan-2-ylpiperazine  
   OTAVA-BB 1194537 
   1-piperidin-4-ylpiperazine 
   4-(Morpholin-4-yl)-piperidine dihydrochloride 
   1-piperidin-4-ylpiperidine;hydrochloride 
   4-cyclohexylpiperidine 
   6-BROMO-2-METHYL-2H-PHTHALAZIN-1-ONE 
   6-chloro-2-methylpyridine-3-carboxylic acid 
   ethyl 6-chloro-2-methylpyridine-3-carboxylate 
   3-bromo-1,5-dimethyl-1,2,4-triazole 
   3-bromo-5-methyl-1H-1,2,4-triazole 
   (3-bromo-1H-1,2,4-triazol-5-yl)methanol 
   methyl 5-bromo-1H-1,2,4-triazole-3-carboxylate 
   2-Azabicyclo[2.1.1]hexane-2,5-dicarboxylicacid2-tertbutylester 
   6-bromo-2H-phthalazin-1-one 
   2-喹啉乙酸 
   6-DIMETHYLAMINO-2-NAPHTHALDEHYDE 
   5-chloropyrido[2,3-d]pyridazine 
   2,6-dichloro-4-cyclopropylpyridine 
   5-pyridin-4-ylpyridin-2-amine 
   5-phenylpyridin-2-amine 
   5-cyclobutylpyridin-2-amine 
   5-cyclopropylpyridin-2-amine 
   METHYL 5-BROMO-3-FLUORO-2-METHYLBENZOATE 
   1,8-NAPHTHYRIDINE-2-CARBOXYLICACIDMONOHYDRATE 
   2-(QUINOLIN-7-YL)ACETIC ACID 
   (R)-TERT-BUTYL 4-(1-AMINOETHYL)PIPERIDINE-1-CARBOXYLATE 
   (S)-TERT-BUTYL 4-(1-AMINOETHYL)PIPERIDINE-1-CARBOXYLATE 
   [1-(aminomethyl)cyclopropyl]methanol 
   6-Amino-3-bromo-2-cyanopyridine 
   TERT-BUTYL N-[(3S,4S)-3-AMINOOXAN-4-YL]CARBAMATE 
   2-chloro-4-isopropylbenzoic acid 
   2-chloro-4-morpholin-4-ylbenzoic acid 
   5-morpholin-4-ylpyridin-2-amine 
   mino-dimethyl-oxo-$l^{6}-sulfane 
   5-ethylpyridin-2-amine 
   5-Difluoromethoxy-pyridin-2-ylamine 
   2-Chloropyrimidine-4-boronicacid 
   1-(2,2-dimethoxyethyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazole 
   2-chloro-4-morpholin-4-ylpyrido[2,3-d]pyrimidine-7-carboxylic acid 
   5,7-dichloro-2-cyclopropylpyrazolo[4,3-d]pyrimidine 
   5,7-Dichloro-1-Methyl-1H-pyrazolo[4,3-d]pyriMidine 
   5,7-dichloro-1H-pyrazolo[4,3-d]pyrimidine 
   3-bromo-7-chloro-2H-pyrazolo[4,3-d]pyrimidine 
   tert-butyl 6-amino-3-azabicyclo[3.1.0]hexane-3-carboxylate 
   TERT-BUTYL 6-FORMYL-3-AZABICYCLO[3.1.0]HEXANE-3-CARBOXYLATE 
   ETHYL ENDO-3-BOC-3-AZABICYCLO-[3.1.0]HEXANE-6-CARBOXYLATE 
   2-Amino-6-(trifluoromethyl)benzoic acid hydrochloride 
   2-Amino-6-(trifluoromethyl)benzoic acid 
   4-Aminobicyclo[2.2.2]octan-1-ol 
   3,6-dihydro-2H-pyran 
   4,7-dioxabicyclo[4.1.0]heptane 
   1-[difluoromethyl(ethoxy)phosphoryl]oxyethane 
   4-chloro-3-iodopyridin-2-amine 
   4-methoxy-2,3-dihydro-1H-isoindole;hydrochloride 
   5-cyclopropyl-3-iodo-1H-pyrazole 
   3-iodo-5-methyl-1H-pyrazole 
   1,5-dimethylpyrazol-3-amine 
   5-bromo-1-methylpyrazolo[3,4-b]pyridine 
   3-methyl-1H-pyrazolo[3,4-b]pyridine-5-carbaldehyde  
   5-bromo-3-ethyl-2H-pyrazolo[3,4-b]pyridine 
   3-ethyl-1H-pyrazolo[3,4-b]pyridine  
   1,3-Dimethyl-1H-pyrazolo[3,4-b]pyridine 
   3-iodo-1-methylpyrazolo[3,4-b]pyridine 
   1-methylpyrazolo[3,4-b]pyridine 
   1H-pyrazolo[3,4-b]pyridine-5-carbonitrile 
   1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid 
   methyl 1H-pyrazolo[3,4-b]pyridine-5-carboxylate 
   5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazolo[3,4-b]pyridine 
   5-iodo-1H-pyrazolo[3,4-b]pyridine 
   1H-pyrazolo[3,4-b]pyridin-5-amine 
   2-fluoro-5-methylpyridine-3-carbaldehyde 
   6-aminopyridine-3-carbaldehyde 
   5-bromo-2-ethylbenzaldehyde 
   5-amino-2-ethoxybenzonitrile 
   5-amino-2-methoxybenzonitrile 
   3-Cyano-4-methoxyphenylboronic acid 
   (3-Cyano-4-isopropoxyphenyl)boronic acid 
   3-cyano-4-ethylphenylboronic acid  
   (3-cyano-4-methylphenyl)boronic acid 
   4-Cyano-3-ethylphenylboronic acid 
   (4-cyano-3-methoxyphenyl)boronic acid 
   (4-Chloro-3-(2-methoxyethoxy)phenyl)boronic acid 
   (4-Chloro-3-propoxyphenyl)boronic acid 
   4-Amino-3-methoxybenzeneboronic acid 
   (3-(Difluoromethoxy)phenyl)boronic acid 
   3-Cyclopropylbenzeneboronic acid  
   (6-phenylpyridin-3-yl)boronic acid 
   4-CYCLOHEXYLPHENYLBORONIC ACID 
   (4-AMINO-3-FLUOROPHENYL)BORONIC ACID 
   4-amino-3-methylphenylboronic acid  
   5-bromo-3-(difluoromethoxy)pyridin-2-amine 
   3-Bromo-5-(difluoromethoxy)pyridine 
   3-bromo-5-pyridin-4-ylpyridine 
   5-Phenyl-3-pyridinyl boronic Acid 
   2-chloro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-3-amine 
   (5-propan-2-yloxypyridin-3-yl)boronic acid 
   5-Ethoxypyridine-3-boronic acid 
   2-Amino-4-(iso-propyl)pyridine 
   3-Pyridinamine, 4-(1-methylethyl)-  
   1-(2,2-dimethylpropyl)piperazine 
   tert-butyl 4-(2,2,2-trifluoroethyl)piperazine-1-carboxylate 
   1-(2,2,2-trifluoroethyl)piperazine 
   1-(pyridin-4-ylmethyl)piperazine 
   1-(cyclopentylmethyl)piperazine 
   1-(cyclopropylmethyl)piperazine 
   1-cyclopropylpiperazine 
   4-(2-bromopyridin-4-yl)morpholine 
   1-(2,2,2-trifluoroethyl)pyrazol-3-amine 
   1-(cyclopropylmethyl)-1H-pyrazol-3-amine 
   1-(Cyclopropylmethyl)-5-iodopyrazole 
   1-(2-methylpropyl)pyrazole 
   1-(2-methylpropyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazole 
   1-(2-methylpropyl)-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazole 
   1-(azidomethyl)-4-methoxybenzene 
   5-bromothiophene-3-carboxylic acid 
   5-(chloromethyl)-2-hydroxybenzaldehyde 
   1,4-Dihydroxynaphthalene 
   (1E,4E)-1,5-di(furan-2-yl)penta-1,4-dien-3-one144850-49-7 
   (E)-6-(4-((4-(trifluoromethoxy)phenyl)diazenyl)phenoxy)hexan-1-ol 
   4-(2-azidoethoxy)benzaldehyde 
   4,4'-(ethane-1,2-diylbis(oxy))dibenzaldehyde 
   4,4',4''-(1,3,5-triazine-2,4,6-triyl)tribenzoic acid 
   3-bromo-9-ethyl-9H-carbazole 
   6-bromo-2-(2-hydroxyethyl)-1H-benzo[de]isoquinoline-1,3(2H)-dione 
   2-(2-aminoethyl)-3',6'-bis(diethylamino)spiro[isoindoline-1,9'-xanthen]-3-one 
   dimethyl 4,4'-((1E,1'E)-(2,5-dimethoxy-1,4-phenylene)bis(ethene-2,1-diyl))dibenzoate 
   3-amino-7-(diethylamino)-2H-chromen-2-one 
   4-ethoxy-3-hydroxybenzaldehyde 
   (E)-2-((phenylimino)methyl)phenol 
   5-(tert-butyl)-2-iodophenol 
   4-(3,4-difluorophenyl)pyrrolidin-2-one 
   (5-(pent-4-en-1-yloxy)pyridin-3-yl)boronic acid 
   1,1,2,2-tetrakis(4-(pyridin-4-yl)phenyl)ethene 
   2-chloro-4-ethoxyphenol 
   4,4',4'',4'''-(ethene-1,1,2,2-tetrayl)tetraaniline 
   2-bromo-4-chloro-6-nitroaniline 
   2-bromo-5-fluoroisonicotinaldehyde 
   1-ethyl-4-vinylbenzene 
   1-bromo-2-fluoro-3-vinylbenzene 
   1-Methyl-3-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole 
   quinolin-5-ol 
   8-chloroquinolin-5-ol 
   1,4-oxathiane 4-oxide 
   2-bromo-7-methoxynaphthalene 
   4-aminoisobenzofuran-1,3-dione 
   4-fluoronicotinic acid 
   3,3-Difluorooxetane 
   2-(trifluoromethyl)cyclopentanone 
   Bis(acetonitrile)dichloropalladium(II) 
   2-amino-5-cyano-3-methylbenzoic acid 
   6-Amino-3-bromo-2-fluorobenzoic acid 
   6-Amino-3-bromopicolinic acid 
   methyl 6-amino-3-bromopyridine-2-carboxylate 
   6-Chloro-4-formylnicotinic acid 
   (3-(2-Cyanopropan-2-yl)phenyl)boronic acid 
   2-methyl-2-(m-tolyl)propanenitrile 
   2-(3-aminophenyl)-2-methylpropanenitrile 
   2-(3-bromophenyl)-2-methylpropanenitrile 
   Benzeneacetonitrile, 2-fluoro-alpha,alpha-dimethyl-  
   METHYL 2-FLUORO-4-METHYL-5-HYDROXYBENZOATE 
   2-Fluoro-5-hydroxy-4-methylbenzoic acid 
   2-Bromo-4-(difluoromethoxy)aniline  
   2-(4-amino-3-chloro-phenyl)-2-methyl-propionitrile 
   2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-5-(trifluoromethoxy)aniline 
   2-Amino-5-morpholinobenzoic Acid 
   Benzoic acid, 2-amino-5-cyclopropyl-  
   5-异丙基邻氨基苯甲酸 
   5-BroMo-4-Fluoro-2-Methylpyridine 
   4-(Difluoromethoxy)-3-nitrobenzoic acid 
   3-Amino-4-cyanobenzoic acid 
   5-iodopyridin-3-amine 
   5-Amino-3-bromo-2-cyanopyridine  
   (3-bromopyridin-4-yl)boronic acid 
   5-Cyclopropylpyridin-3-ylboronic acid 
   (5-Morpholinopyridin-3-yl)boronic acid 
   3-Bromo-4-(difluoromethoxy)pyridine 
   1-cyclobutylpiperazine 
   1-cyclopropyl-3,3-bis(methylthio)propan-1-one 
   1-cyclohexyl-3,3-bis(methylthio)propan-1-one 
   2-Propen-1-one, 3,3-bis(methylthio)-1-(4-pyridinyl)-  
   3,3-bis(methylsulfanyl)-1-pyridin-2-ylprop-2-en-1-one 
   3,3-bis(methylsulfanyl)-1-phenylprop-2-en-1-one 
   3-Pyridinecarboxylicacid,5-ethyl-(9CI) 
   5-Morpholinonicotinic acid 
   5-(Piperidin-1-yl)nicotinic acid 
   5-pyridin-3-ylpyridine-3-carboxylic acid 
   5-phenylpyridine-3-carboxylic acid 
   5-Cyclopropylnicotinic acid 
   3-Pyridinecarboxylicacid,5-(1-methylethyl)-(9CI) 
   5-(difluoromethoxy)pyridin-3-ylboronic acid 
   3-Bromo-5-(difluoromethoxy)pyridine 
   2-chloro-3-(difluoromethoxy)pyridine 
   3-iodocyclopent-2-en-1-one 
   (3R,4S)-1-BOC-3-FLUORO-4-HYDROXYPYRROLIDINE 
   3-cyclobutyl-1H-pyrazole-5-carboxylic acid 
   3-cyclobutyl-1H-pyrazole 
   3-Fluoro-1H-pyrazole 
   1-(tert-butyl)-3,5-dimethyl-1H-pyrazole 
   7-Chloro-naphthalene-1-carboxylic acid 
   7-Bromo-1-naphthoic acid 
   (5-bromo-1-benzothiophen-3-yl)methanamine;hydrochloride 
   3-bromo-5,6,7,8-tetrahydro-1,7-naphthyridine 
   Methyl 3,?4-?dihydro-?1H-?2-?benzopyran-?1-?acetate 
   1-?Chloro-?3,?4-?dihydro-?1H-?2-?benzopyran 
   2-?(3-?chloropyridin-?4-?yl)?acetic acid 
   3-CHLOROPYRIDINE-2-ACETIC ACID 
   TERT-BUTYL 3-FLUORO-4-OXOPYRROLIDINE-1-CARBOXYLATE 
   tert-butyl 3-bromo-4-oxopyrrolidine-1-carboxylate 
   1-methylpiperazin-2-one 
   (4-(Difluoromethoxy)-3-fluorophenyl)boronic acid 
   (4-aminophenyl)-(4-hydroxyphenyl)methanone 
   methyl 2-methyloxazole-5-carboxylate 
   环丙硫醇钠 
   tert-Butyl oxazol-5-ylcarbamate 
   1,3-oxazol-5-amine 
   piperidine-2,3-dione 
   3-hydroxypiperidin-2-one 
   tert-?butyl N-?{2-?[(1-?methyl-?1H-?pyrazol-?4-?yl)?methyl]?-?3-?oxopropyl}?carbamate 
   3,4-DIHYDRO-2H-1,4-BENZOXAZINE-2-CARBOXYLIC ACID 
   tert-butyl N-benzyl-N-(2-hydroxyethyl)carbamate 
   2-methylindazole-4-carbaldehyde 
   2,4-dimethyl-2H-indazole 
   3-methyl-1,2-oxazole-4-carboxylic acid 
   2-bromo-1,3,4-Oxadiazole 
   3-Bromopyrazine-2-carbaldehyde 
   8-bromo-[1,2,4]triazolo[4,3-a]pyridine 
   7-amino-2,3-dihydroinden-1-one 
   tert-butyl 4-(2,2,2-trifluoroethyl)piperazine-1-carboxylate 
   1-(2,2,2-trifluoroethyl)piperazine 
   1-(2,2-difluoroethyl)piperazine 
   3-cyclohexyl-3-oxopropanenitrile 
   5-cyclohexyl-1H-pyrazol-3-amine 
   3-cyclobutyl-3-oxopropanenitrile 
   5-cyclobutyl-1H-pyrazol-3-amine 
   2,6-Difluoropyridine-4-boronic acid 
   2,6-Dichloropyridine-4-boronic acid 
   3-(4-fluorophenyl)pyrrolidine 
   3-(3-fluorophenyl)pyrrolidine 
   3-(3-chlorophenyl)pyrrolidine 
   3-(3-bromophenyl)pyrrolidine 
   3-(3-methoxyphenyl)pyrrolidine 
   5-iodo-2,2-dimethylpentanenitrile 
   5-chloro-2,2-dimethylpentanenitrile 
   pyrido[3,2-d]pyridazin-8(7H)-one 
   2-chloro-6-cyclobutylBenzoic acid 
   4-Chloro-3-isopropylbenzoic acid 
   3-Chloro-[1,1'-biphenyl]-4-carboxylic acid 
   5-bromo-8-methoxyquinazoline 
   5-bromo-3-cyclopropyl-2H-pyrazolo[3,4-b]pyridine 
   1H-Pyrazolo[3,4-b]pyridine, 5-bromo-3-phenyl- 
   3-Phenyl-7-aza-1H-indazloe 
   2-(3-bromo-4-fluorophenyl)-2-methylpropanenitrile 
   3-Methyl-1H-pyrazolo[3,4-b]pyridine-5-boronic acid pinacol ester 
   PYRAZOLO[1,5-A]PYRIDIN-5-OL 
   6,7-dimethyl-quinoline-4-carboxylic acid 
   6-chloro-3-iodopyridin-2-ol 
   6-Chloro-5-(trifluoromethyl)nicotinonitrile 
   tert-butyl (1S,2R)-2-aminocyclohexylcarbamate 
   3,3-dichloro-4-hydroxy-butan-2-one 
   6-Fluoro-1,2,3,4-Tetrahydro-Isoquinoline 
   6-Fluoro-1,2,3,4-Tetrahydro-Isoquinoline Hydrochloride 
   2-Pyridineaceticacid 
   6-bromo-5-methoxypyridin-2-amine 
   3-(2-Chloro-phenyl)-pyrrolidine 
   4-bromo-5-methyl-1H-indazole 
   1-[(tert-butoxy)carbonyl]-3-fluoroazetidine-3-carboxylic acid 
   methyl (S)-2-(5-(bromomethyl)-2-chlorophenoxy)propanoate 
   4-bromobenzenesulfonic acid hydrate 
   N-(3,4-Dimethyl-5-isoxazolyl)-N-sulfanilylacetamide 
   2-BROMO-6-ISOPROPYL-ANILINE 
   7-Benzyl-5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine-1-carboxylic acid ethyl ester 
   8-Methoxy-isochroman 
   5-Fluoro-pyrimidine-2-carboxylic acid ethyl ester 
   5-Chloro-pyrimidine-2-carboxylic acid ethyl ester 
   3-Aza-bicyclo[3.2.1]octan-8-ol 
   2,2,2-Trifluoro-N-pyrimidin-2-yl-acetamide 
   8-Carboxymethyl-3-aza-bicyclo[3.2.1]octane-3-carboxylic acid tert-butyl ester 
   6,6-Difluoro-2-aza-bicyclo[2.2.1]heptane 
   (5-Bromo-pyrimidin-2-yl)-acetic acid methyl ester 
   7H-Pyrrolo[2,3-d]pyrimidin-2-ylamine 
   6-Hydroxy-2-aza-bicyclo[2.2.1]heptane-2-carboxylic acid tert-butyl ester 
   (8-Oxa-bicyclo[3.2.1]oct-3-yl)-carbamic acid tert-butyl ester 
   3-Bromo-4-chloro-3H-pyrazolo[3,4-d]pyrimidine 
   8-Aza-bicyclo[3.2.1]octane-2-carboxylic acid 
   3-Iodo-imidazo[1,5-a]pyrazine 
   7-Bromo-6-chloro-8-fluoro-quinazolin-4-ol 
   5-Bromo-6-chloro-pyridazin-3-ol 
   3-Adamantan-1-yl-2-amino-propionic acid 
   6-(1-Acetyl-piperidin-4-ylamino)-pyrimidine-4-carboxylic acid 
   2,6-二溴苯甲醚 
   2-溴4-氟三氟甲苯 
   2-氨基-5-甲氧基三氟甲苯 
   2.6-二氟-4-溴碘苯 
   2-硝基-3.5二氟苯酚 
   2.5-二溴苯酚 
   2,3-二甲基-4-氟硝基苯 
   2-氟-6-碘硝基苯 
   2-碘-3-溴硝基苯 
   3-氟-4-溴苯乙腈 
   2-甲基-4-甲氧基苯甲酸甲脂 
   5-氟-2-溴苯睛 
   2,3-二氟-6-溴苯睛 
   3-氟-5-溴苯甲醛 
   2.3-二氟苯甲醛 
   2-氟-6-甲基苯甲醛 
   2-氟-4-三氟甲基苯甲醛 
   2-氟-4-碘苯甲醛 
   2-甲氧基-5-氟苯甲醛 
   3-三氟甲基-5-甲氧基苯甲醛 
   3-氟-4-氰基苯甲醛 
   3-氟-5-氰基苯甲醛 
   2-氟-3-氯苯乙酮 
   2-氟-6-氯苯乙酮 
   2-溴-4-氯苯乙酮 
   2-氟-6-溴苯乙酮 
   3-氟-4-溴苯乙酮 
   2,3,6-三氟苯乙酸 
   3-氯-2.6-二氟苯甲酸 
   3-羟基-5-三氟甲基苯甲酸 
   5-溴-2.4-二氟苯甲酸 
   2-碘-5-硝基苯甲酸甲脂 
   4-氟-3-羟基苯甲酸 
   2-甲基-3.4-二氟苯甲酸 
   2-氟-5-羟基苯甲酸 
   2-氨基-5-三氟甲基苯甲酸 
   3-氟-2-硝基苯甲酸 
   2-氟-4-碘苯甲酸 
   2-氨基-45-二氯苯甲酸 
   2-溴-4-氟硝基苯 
   26-二溴氟苯 
   3-氟-5-碘苯甲酸 
   2-甲基-4-溴-5-氟苯腈 
   3-溴-2氟苯胺 
   24-二氟-5-氯硝基苯 
   2-氰基-5-氟溴苄 
   26-二氯-4-氟苯胺 
   3-羟基-4-溴苯甲酸甲脂 
   26-二溴氯苯 
   2-氟-4-氰基苯甲酸 
   2-氰基-5-氟苯甲酸甲脂 
   2-氨基-5-甲氧基苯甲酸甲脂 
   35-二氟-4-氰基苯甲醛 
   3-溴-2-氯三氟甲苯 
   35-二碘-4-羟基苯甲醛 
   34-二溴硝基苯 
   26-二氟-4-溴硝基苯 
   35-二氟-4-氨基苯甲酸 
   2-碘-4-甲氧基苯甲酸 
   2-溴-4-氟硝基苯 
   35-二甲基-4-溴苯腈 
   345-三苄氧基苯甲酸甲脂 
   26-二氟碘苯 
   3-溴-12-二氨基苯 
   24-二氟-3-甲氧基苯甲酰胺 
   35-二氟-4-氯苯腈 
   2-氯-3-氟-5-溴苯甲醚 
   2-氯-3-氟-5-溴苯酚 
   24-二氟-5-氯苯胺 
   2-溴-46-二氟苯胺 
   35-二氟-4-溴苯甲酸 
   2-氟-6-羟基苯甲醛 
   2-氯-4-甲氧基苯胺 
   2-胺基-5-硝基苯甲酸甲脂 
   3甲基-4-碘苯甲酸甲脂 
   26-二氟-4-溴苯腈 
   3-溴-2-氟苯甲酸甲脂 
   26-二氟-4-溴苯甲酸 
   2-甲氧基-4-溴-5-氟苯胺 
   24-二氟-5-溴硝基苯 
   2-氟-5-羟基苯甲酸甲脂 
   2-氯-35-二氟溴苯 
   25-二氟-4-溴苯腈 
   2-溴-4-氟-5-氯硝基苯 
   35-二氟碘苯 
   246-三氟苯甲酸 
   2-氯-4-氟-5-硝基苯甲醚 
   2-胺基-35-二氟苯腈 
   2-氟-6-羟基苯甲酸甲酯 
   2-氯-4-氟-5-溴硝基苯 
   2-氟-5-羟基苯腈 
   3-苄氧基溴苯 
   3-氟-5-溴苯甲酸甲酯 
   25-二氟-4-溴苯甲酸 
   2-胺基-35-二氟苯甲酸 
   2-甲基-6-溴苯胺 
   2-胺基-3-氯-4-氟硝基苯 
   2-羟基-4-氟苯腈 
   2-氟-4-溴-5-硝基苯甲醚 
   24-二甲基溴苄 
   2-氟-5-甲氧基苯胺 
   2-溴-4-甲基-5-氟苯甲醛 
   2-甲氧基-4-胺基苯腈 
   2-碘-5-氟苯乙酮 
   3-甲氧基-4-溴苯甲酸 
   2-甲基-4-氟苯腈 
   3-甲氧基-4-溴苯腈 
   4-异丙基-2-硝基甲苯 
   3-甲氧基-5-溴苯甲酸 
   3-溴-4-三氟甲基苯甲酸 
   345-三氟苯乙腈 
   24-二氟苯乙腈 
   35-二甲氧基氟苯 
   3-甲氧基-4-氟苯腈 
   2-溴-5-氯硝基苯 
   2-三氟甲基-4-碘苯甲酸 
   2-氟-5-氰基苯甲酸 
   2-三氟甲基-4-硝基苯甲酸甲酯 
   3-溴-2-氯苯胺 
   2-氨基-4-硝基苯腈 
   2-氟-6-三氟甲基苯腈 
   3-溴-2-氟硝基苯 
   2-氟-6-溴硝基苯 
   2-氯-4-溴苯胺 
   2-硝基-45-二氟苯甲酸 
   2-溴-35-二氟苯甲酸 
   2-溴-3-氟三氟甲苯 
   2-氟-4-溴苯乙酮 
   2-氨基-6-溴苯甲酸  
   2-氨基-6-溴苯甲酸 盐酸盐 
   26-二甲基-4-氯溴苯 
   24-二氟-6-甲氧基硝基苯 
   35-二氟-4-硝基苯腈 
   3-溴-2-氨基硝基苯 
   3-硝基-4-氟苯甲醚 
   3-溴-5-胺基苯甲酸 
   26-二氟-3-溴苯甲酸 
   2-甲氧基-4-氟苯腈 
   2-甲氧基--4-氟硝基苯 
   2-氯-4-硝基三氟甲苯 
   246-三溴甲苯 
   Methyl 4-(aminomethyl)benzoate 
   (4-(1-morpholinoethyl)phenyl)boronic acid hydrochloride 
   [4-[(4-Methyl-1-piperazinyl)sulfonyl]phenyl]boronic acid 
   B-[4-[1-(1-Pyrrolidinyl)ethyl]phenyl]boronic acid 
   [4-(N-Cyclopropylaminocarbonyl)phenyl]boronic acid 
   5-phenyl-1H-1,2,4-triazol-3-amine 
   4-bromo-3-hydroxybenzaldehyde 
   1-(bromomethyl)-2-methoxybenzene 
   3-Bromostyrene 
   3-Aminomethylbenzoic acid hydrochloride 
   5-Methylthiazole-4-carboxylic acid 
   Ethyl 5-bromothiazole-4-carboxylate 
   3-vinylaniline 
   4-Bromopyrimidine hydrobromide 
   5-Hexenylboronic acid 
   2-(2-bromoethoxy)tetrahydro-2H-pyran 
   Cyanocyclobutane 
   5-bromopyrimidin-4-amine 
   (1S,2R)-2-(tert-butoxycarbonylamino)cyclopentanecarboxylic acid 
   1-(3-bromophenyl)imidazolidin-2-one 
   2-hydrazinylpyrazine 
   2-iodopyrazine 
   pyridazine-3,6-diamine 
   propan-2-amine hydrochloride 
   4-Hydroxy-3-methoxystyrene 
   2-fluoropyrazine 
   methyl 1H-indazole-6-carboxylate 
   4-(trifluoromethyl)pyrimidin-2-amine 
   5-bromo-4-(trifluoromethyl)pyrimidin-2-amine 
   6-bromo-5-methyl-1H-indazole 
   5-bromo-6-methyl-1H-indazole 
   2-(methylsulfonyl)acetic acid 
   1,7-naphthyridin-8-amine 
   2-Amino-5-bromobenzothiazole 
   2-aminonicotinamide 
   2-Cyano-5-nitropyridine 
   4-(5-Nitropyridin-2-yl)morpholine 
   10-hydroxy-10,11-dihydro-5H-dibenzo[b,f]azepine-5-carboxamide 
   pyridazine-4,5-dicarboxylic acid 
   7-bromo-2-methyloxazolo[4,5-c]pyridine 
   2-(2-bromophenyl)-1,3-dioxolane 
   methyl 4-(aminomethyl)benzoate hydrochloride 
   2-aminobenzo[d]thiazol-6-ol 
   2-(hydroxymethyl)benzoic acid 
   3,6-Diiodopyridazine 
   2-ethyl-1,3,4-oxadiazole 
   3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)pyridine 
   (4-(trifluoromethyl)pyridin-3-yl)boronic acid 
   2-isopropoxy-5-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-3-(trifluoroMethyl)pyridine 
   N-ethyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-3-(trifluoromethyl)pyridin-2-amine 
   N-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-3-(trifluoromethyl)pyridin-2-amine 
   2-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-3-(trifluoromethyl)pyridine 
   2-Benzyloxy-5-(trifluoromethyl)pyridine-3-boronic acid 
   5-Trifluoromethyl-pyridine-3-boronic acid 
   (6-(2,4-dichlorophenoxy)pyridin-3-yl)boronic acid 
   6-(2-Morpholinoethoxy)pyridine-3-boronic acid 
   6-(4-(trifluoromethoxy)phenoxy)pyridin-3-ylboronic acid 
   2-(4-TrifluoroMethylphenoxy)pyridine-5-boronic acid 
   (6-(3,4-difluorophenoxy)pyridin-3-yl)boronic acid 
   6-ethoxy-5-(trifluoroMethyl)pyridin-3-ylboronic acid 
   (6-(2-fluorophenoxy)pyridin-3-yl)boronic acid 
   6-(benzyloxy)-5-Methylpyridin-3-ylboronic acid 
   (6-((tetrahydro-2H-pyran-4-yl)methoxy)pyridin-3-yl)boronic acid 
   (6-((4-fluorobenzyl)oxy)pyridin-3-yl)boronic acid 
   (6-((4-chlorobenzyl)oxy)pyridin-3-yl)boronic acid 
   (6-(4-cyclopropylphenoxy)pyridin-3-yl)boronic acid 
   (6-(3-fluorophenoxy)pyridin-3-yl)boronic acid 
   6-(Tetrahydropyran-4-yloxy)pyridine-3-boronic acid 
   6-(4-Methoxybenzyloxy)pyridin-3-ylboronic acid 
   (6-(4-fluorophenoxy)pyridin-3-yl)boronic acid 
   (6-(dodecyloxy)pyridin-3-yl)boronic acid 
   (6-phenethoxypyridin-3-yl)boronic acid 
   (6-(cyclohexyloxy)pyridin-3-yl)boronic acid 
   (6-(4-methoxyphenoxy)pyridin-3-yl)boronic acid 
   6-(cyclopentyloxy)pyridine-3-boronic acid 
   (6-(hexyloxy)pyridin-3-yl)boronic acid 
   (2-isopropyl-6-methoxypyridin-3-yl)boronic acid 
   (6-(pentyloxy)pyridin-3-yl)boronic acid 
   2-Phenoxypyridin-5-yl boronic acid hydrochloride 
   (2-ethyl-6-methoxypyridin-3-yl)boronic acid 
   (6-butoxypyridin-3-yl)boronic acid 
   (6-ethoxy-5-methylpyridin-3-yl)boronic acid 
   4,6-Dimethoxypyridine-3-boronic acid 
   2,6-Dimethoxypyridine-3-boronic acid 
   (6-(difluoromethoxy)pyridin-3-yl)boronic acid 
   2-Propoxypyridine-5-boronic acid 
   (6-methoxy-2-methylpyridin-3-yl)boronic acid 
   6-Methoxy-4-methylpyridine-3-boronic acid;Boronic acid 
   2-fluoro-6-(methylamino)pyridin-3-ylboronic acid 
   (6-(dimethylamino)-5-fluoropyridin-3-yl)boronic acid 
   5-fluoro-6-Morpholinopyridin-3-ylboronic acid 
   2-Benzyloxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-(2-methoxyethoxy)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-(difluoromethoxy)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2,6-dimethoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-isopropoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-ethoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-Methoxy-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-chloro-6-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-chloro-3-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-chloro-5-fluoro-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2,6-dichloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-methoxy-6-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-cyclopropyl-6-methyl-4-(4,4,5,5,-tetramethyl-1,3,2-dioxa-borolan-2-yl)-pyridine 
   6-Methyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)picolinonitrile 
   2-Bromo-6-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-chloro-6-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2,5-Dimethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-pyridine 
   4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-2-pyridinecarbonitrile 
   2,6-dimethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-fluoro-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-6-(trifluoroMethyl)pyridine 
   2-bromo-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-6-(trifluoromethyl)pyridine 
   4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)pyridine 
   2-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-6-(trifluoromethyl)pyridine 
   2-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-6-(trifluoromethyl)pyridine 
   N,N-diethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinamide 
   tert-butyl 6-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate 
   ethyl 6-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate 
   N,N-dimethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinamide 
   ethyl 4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)picolinate 
   methyl 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate 
   (6-(4-methylpiperidin-1-yl)pyridin-3-yl)boronic acid 
   (6-(4-(tert-butoxycarbonyl)piperazin-1-yl)pyridin-3-yl)boronic acid 
   (6-(4-ethylpiperazin-1-yl)pyridin-3-yl)boronic acid 
   (6-(4-methylpiperazin-1-yl)pyridin-3-yl)boronic acid 
   (6-(Piperidin-1-yl)pyridin-3-yl)boronic acid 
   6-pyrrolidin-1-yl- pyridineboronic acid 
   6-(tert-Butoxycarbonyl(methyl)amino)pyridin-3-ylboronic acid 
   (6-(methylamino)pyridin-3-yl)boronic acid 
   2-(Dimethylamino)pyridine-5-boronic acid hydrate 
   methyl 1H-pyrrolo[3,2-c]pyridine-6-carboxylate 
   methyl 5-bromo-1H-indazole-4-carboxylate 
   methyl 5-bromo-1H-indazole-4-carboxylate 
   5-Trifluoromethyl-pyridin-3-ylamine 
   (1,5-dimethyl-1H-imidazol-2-yl)methanol 
   Methyl 3-aMino-2-(aMinoMethyl)propanoate dihydrochloride 
   5-bromo-7H-pyrrolo[2,3-d]pyrimidin-2-amine 
   2,4-Dichloro-5-methyl-7H-pyrrolo[2,3-d]pyrimidine 
   6-bromo-4-chlorothieno[2,3-d]pyrimidine 
   2,6-dichloroquinazoline 
   7-(trifluoromethyl)quinazoline-2,4(1H,3H)-dione 
   Methyl imidazo[1,2-b]pyridazine-6-carboxylate 
   methyl 5-methoxypyrimidine-2-carboxylate 
   Imidazo[1,2-a]pyridin-6-amine 
   4-(methoxycarbonyl)cubane-1-carboxylic acid 
   Bicyclo[1.1.1]pentane-1,3-dicarboxylic acid 
   (1S,3R,4S)-2-(Tert-Butoxycarbonyl)-2-Azabicyclo[2.2.2]Octane-3-Carboxylic Acid 
   2-Chloropyrimidine-5-carboxylic acid 
   exo-3-Boc-aminotropane 
   tert-Butyl 4-chloro-5H-pyrrolo[3,4-d]pyrimidine-6(7H)-carboxylate 
   endo-3-Boc-aminotropane 
   5-Chloro-2-cyanopyrazine 
   4-(Benzyloxy)cyclohexanone 
   4-Chloro-1,8-dimethyl-imidazo[1,2-a]quinoxaline 
   2,2-Diphenylethylenone 
   2,7-Naphthyridine-3-carboxylic acid 
   7-Bromo-1,2,3,4-tetrahydroquinoline 
   6-Methylpyridazin-3-amine 
   3-amino-5-chloro-[1,1'-biphenyl]-4-ol 
   3-chloro-5-nitro-[1,1'-biphenyl]-4-ol 
   4-(chloromethyl)-3-iodopyridine 
   3-iodoisonicotinaldehyde 
   3-propoxybenzonitrile 
   (3-iodopyridin-4-yl)methanol 
   4-(3,4,5-trifluorophenyl)pyrrolidin-2-one 
   (S)-4-(3,4,5-trifluorophenyl)pyrrolidin-2-one 
   (R)-4-(3,4,5-trifluorophenyl)pyrrolidin-2-one 
   4,6-dichloro-1H-pyrazolo[3,4-b]pyridine 
   (2-(aminomethyl)phenyl)boronic acid hydrochloride 
   5-Chloro-6-ethylpyrimidin-4-amine 
   tert-butyl (S)-3-(4-bromophenyl)piperidine-1- carboxylate 
   trans-N-[1-(2-Fluorphenyl)-1H-pyrazol-3-yl]-1’-oxospiro[cyclohexane-1,3’(1’H)-furo[3,4-c]pyridine]-4-carboxamide;(1r,4r)-N-(... 
   N-(4-isopropoxyphenyl)-4-(6-methoxy-7-(3-(piperidin-1-yl)propoxy)quinazolin-4-yl)piperazine-1-carboxamide 
   (R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 
   N-[5-(4-Bromophenyl)-6-[2-[(5-bromo-2-pyrimidinyl)oxy]ethoxy]-4-pyrimidinyl]-N'-propylsulfamide 
   (R)-2-[[6-(3-AMinopiperidin-1-yl)-3-Methyl-2,4-dioxo-3,4-dihydropyriMidin-1(2H)-yl]Methyl]-4-fluorobenzonitrile 
   ApreMilast, (S)-2-[1-(3-Ethoxy-4-Methoxyphenyl)-2-Methylsulfonylethyl]-4-acetylaMinoisoindoline-1,3-dione 
   methyl (3Z)-3-[[4-[methyl-[2-(4-methylpiperazin-1-yl)acetyl]amino]anilino]-phenylmethylidene]-2-oxo-1H-indole-6-carboxylate 
   (3Z)-2,3-Dihydro-3-[[[4-[methyl[2-(4-methyl-1-piperazinyl)acetyl]amino]phenyl]amino]phenylmethylene]-2-oxo-1H-indole-6-carbo... 
   β-D-Fructopyranose;(S)-3-methyl-2-((((2S,3S,4R,5R)-2,3,4,5-tetrahydroxytetrahydro-2H-pyran-2-yl)methyl)thio)butanoic acid 
   (1S,4R,5S,6R)-4,5,6-trihydroxy-3-(hydroxymethyl)cyclohex-2-en-1-yl dihydrogen phosphate 
   N-Octanoyl-D-erythro-sphingosine;N-((2S,3R,E)-1,3-dihydroxyoctadec-4-en-2-yl)heptanamide 
   D-erythro-sphingosine;(2S,3R,E)-2-aminooctadec-4-ene-1,3-diol 
   2-(1-(4,4-difluorocyclohexyl)piperidin-4-yl)-6-fluoro-3-oxoisoindoline-4-carboxamide 
   6-(4-amino-4-methylpiperidin-1-yl)-3-(2,3-dichlorophenyl)pyrazin-2-amine hydrochloride 
   (R)-9-(1-acryloylpiperidin-3-yl)-6-amino-7-(4-phenoxyphenyl)-7H-purin-8(9H)-one 
   (R)-6-amino-9-(1-but-2-ynoylpyrrolidin-3-yl)-7-(4-phenoxyphenyl)-7H-purin-8(9H)-one HCl salt 
   Methyl 1-(4-bromophenyl)cyclopropanecarboxylate 
   1-(4-Bromophenyl)cyclopropanecarbonitrile 
   7-Bromopyrido[2,3-b]pyrazine 
   2-(4,4-Difluoropiperidin-1-yl)ethanamine 
   [1,2,4]Triazolo[1,5-a]pyridin-7-ylboronic acid 
   4-(4-Hydrazinylbenzyl)oxazolidin-2-one 
   Methyl 4-amino-1-methyl-1H-imidazole-2-carboxylate 
   (S)-3-(1-(Dimethylamino)ethyl)phenyl ethyl(methyl)carbamate 
   Dimethyl (4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)phosphonate 
   1,3-Diiodobenzene 
   1,4-Diiodobenzene 
   1-Bromo-4-iodobenzene 
   (4-Bromophenyl)boronic acid 
   (2,3-Dimethylphenyl)boronic acid 
   (4-(Diphenylamino)phenyl)boronic acid 
   2-([1,1':4',1''-Terphenyl]-4-yl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 
   Phenanthren-9-ylboronic acid 
   (3-(Naphthalen-1-yl)phenyl)boronic acid 
   (4-(Naphthalen-1-yl)phenyl)boronic acid 
   [1,1'-Biphenyl]-3-ylboronic acid 
   Benzenesulfonic thioanhydride 
   2,7-Dibromo-9H-fluorene 
   9,10-Dibromoanthracene 
   Potassium 4,6-dioxo-1,4,5,6-tetrahydro-1,3,5-triazine-2-carboxylate 
   (S)-2-Phenyloxirane 
   2-(4-Bromo-1H-indol-3-yl)acetonitrile 
   2-Cyclopropyl-6-oxo-1,6-dihydropyrimidine-4-carboxylic acid 
   (1R,2S)-2-((tert-butoxycarbonyl)amino)cyclopentanecarboxylic acid 
   (S)-2-(Benzylamino)-1-phenylethanol 
   Methyl 3-bromo-2-nitrobenzoate 
   2-(Methylsulfonyl)-5-(trifluoromethyl)-1,3,4-thiadiazole 
   (3-Bromo-2-methoxyphenyl)methanol 
   2-Chloro-5-vinylpyrimidine 
   4-Iodo-1H-indole 
   2,6-Dichloro-4-iodophenol 
   3,4-Dinitrophenol 
   2-Bromo-5-fluoro-4-(trifluoromethyl)pyridine 
   1,3-Dibromo-2-methyl-propane 
   5-Bromo-2-methylpyridin-4-amine 
   4-(Azetidin-1-yl)piperidine 
   ethyl 1-(4-bromophenyl)-5-methyl-1H-1,2,3-triazole-4-carboxylate 
   1-(4-Bromophenyl)-5-methyl-1H-1,2,3-triazole-4-carboxylic acid 
   Bicyclo[3.2.1]octane-2,4-dione 
   Imidodisulfuryl fluoride lithium salt 
   (3-Bromo-5-chloropyridin-4-yl)methanol 
   4-Chloro-5H-pyrrolo[3,2-d]pyrimidine 
   4,4'-Di-tert-butyl-2,2'-bipyridine 
   (Bromomethyl)cyclopentane 
   1H-Pyrrolo[2,3-b]pyridine-4-carbonitrile 
   Sodium 2-methylpropane-2-thiolate 
   4-Bromo-1-cyclopropyl-1H-pyrazole 
   (2S,3S)-Methyl 2-aMino-3-hydroxybutanoate hydrochloride 
   Basmisanil 
   Pyridine,compd.withsulfurtrioxide(1:1) 
   1,4-BUTANEDIOL-D10 
   ADIPIC-D8 ACID-D2 
   8-Bromo-3,4-dihydro-1H-benzo[e][1,4]diazepin-5(2H)-one 
   Methyl 4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-yl)benzoate 
   Dimethyl 5-(bromomethyl)isophthalate 
   4-(Aminomethyl)benzimidamide dihydrochloride 
   (S)-1-(tert-Butoxycarbonyl)piperazine-2-carboxylic acid 
   (4-Octylphenyl)boronic acid 
   (4-(Decyloxy)phenyl)boronic acid 
   Propane-1-sulfonamide 
   2-Ethyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxylic acid 
   6-Chloro-1-methyl-1H-imidazo[4,5-c]pyridine 
   4-(((tert-Butoxycarbonyl)amino)methyl)picolinic acid 
   2-Methylbenzo[d]thiazol-7-amine 
   (4-((tert-butyldimethylsilyl)oxy)-3-fluorophenyl)boronic acid 
   (3-((4-((tert-butyldiphenylsilyl)oxy)piperidin-1-yl)sulfonyl)phenyl)boronic acid 
   (3-((4-(2-((tert-butyldiphenylsilyl)oxy)ethyl)piperazin-1-yl)sulfonyl)phenyl)boronic acid 
   (4-(1-(piperazin-1-yl)ethyl)phenyl)boronic acid 
   (3-((4-(2-hydroxyethyl)piperazin-1-yl)sulfonyl)phenyl)boronic acid 
   (3-(N-(tert-butyl)sulfamoyl)phenyl)boronic acid 
   (3-(N-cyclopentylsulfamoyl)phenyl)boronic acid 
   (5-((4-hydroxypiperidin-1-yl)sulfonyl)-2-methylphenyl)boronic acid 
   (3-(aminomethyl)phenyl)boronic acid hydrochloride 
   potassium trifluoro(3-oxo-3-(pyrrolidin-1-yl)propyl)borate 
   potassium trifluoro(3-(4-methylpiperidin-1-yl)-3-oxopropyl)borate 
   (3-((2,5-dimethoxyphenyl)amino)-3-oxopropyl)trifluoroborate 
   potassium (3-((4-bromo-2-fluorophenyl)amino)-3-oxopropyl)trifluoroborate 
   potassium (3-((5-bromo-2-fluorophenyl)amino)-3-oxopropyl)trifluoroborate 
   potassium (3-((3-bromo-4-fluorophenyl)amino)-3-oxopropyl)trifluoroborate 
   potassium (3-((3-chloro-4-fluorophenyl)amino)-3-oxopropyl)trifluoroborate 
   potassium trifluoro(3-((2-nitrophenyl)amino)-3-oxopropyl)borate 
   (2-fluoro-5-(N-isopropylsulfamoyl)-4-methylphenyl)boronic acid 
   N-cyclohexyl-2-(4-(4,4,5,5-tetramethyl-1,3-dioxolan-2-yl)phenoxy)acetamide 
   (3-fluoro-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)boronic acid 
   (4-(2-(4-methylpiperazin-1-yl)ethoxy)phenyl)boronic acid 
   (5-((4-ethylpiperazin-1-yl)sulfonyl)-2-methylphenyl)boronic acid 
   (5-(N,N-diethylsulfamoyl)-2-methylphenyl)boronic acid 
   (2-methyl-5-(piperazin-1-ylsulfonyl)phenyl)boronic acid 
   (5-((4-(tert-butoxycarbonyl)piperazin-1-yl)sulfonyl)-2-methylphenyl)boronic acid 
   N-isopropyl-2-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenoxy)acetamide 
   (4-(3-(cyclohexylamino)propoxy)-3-fluorophenyl)boronic acid hydrochloride 
   (4-(N-(tert-butyl)sulfamoyl)-3,5-dimethylphenyl)boronic acid 
   (2-(hydroxymethyl)-4-methoxyphenyl)boronic acid 
   (4-(N-isopropylsulfamoyl)-3,5-dimethylphenyl)boronic acid 
   (4-(N-(4-methoxybenzyl)sulfamoyl)-3,5-dimethylphenyl)boronic acid 
   (4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-2-fluorophenyl)boronic acid 
   (5-(N,N-diethylsulfamoyl)-2-fluorophenyl)boronic acid 
   (2-fluoro-4-((4-oxopiperidin-1-yl)methyl)phenyl)boronic acid 
   N-(2-fluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-2-(4-methylpiperidin-1-yl)acetamide 
   2-(4-ethylpiperazin-1-yl)-N-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acetamide 
   2-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 
   2-(4-methylpiperazin-1-yl)-N-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acetamide 
   (4-(N-cyclopropylsulfamoyl)-2,5-difluorophenyl)boronic acid 
   2-chloro-N-(4-fluoro-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acetamide 
   (3-(N,N-diethylsulfamoyl)-4-fluorophenyl)boronic acid 
   (3-(N-cyclopropylsulfamoyl)-4-fluorophenyl)boronic acid 
   potassium ((dimethylamino)methyl)trifluoroborate 
   (3-(N,N-dimethylsulfamoyl)-4-fluorophenyl)boronic acid 
   (4-fluoro-3-(pyrrolidin-1-ylsulfonyl)phenyl)boronic acid 
   (4-fluoro-3-(morpholinosulfonyl)phenyl)boronic acid 
   (2-fluoro-4-methyl-5-(N-methylsulfamoyl)phenyl)boronic acid 
   potassium ((cyclohexylamino)methyl)trifluoroborate 
   (5-((4-ethylpiperazin-1-yl)sulfonyl)-2-fluoro-4-methylphenyl)boronic acid 
   4-fluoro-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 
   (2-fluoro-4-methyl-5-((4-methylpiperazin-1-yl)sulfonyl)phenyl)boronic acid 
   (5-(N-cyclopropylsulfamoyl)-2-fluoro-4-methylphenyl)boronic acid 
   (5-(N,N-dimethylsulfamoyl)-2-fluoro-4-methylphenyl)boronic acid 
   (2-fluoro-4-methyl-5-((4-methylpiperidin-1-yl)sulfonyl)phenyl)boronic acid 
   (5-chloro-6-(dimethylamino)pyridin-3-yl)boronic acid 
   (5-(N,N-diethylsulfamoyl)-2-fluoro-4-methylphenyl)boronic acid 
   (5-chloro-6-(pyrrolidin-1-yl)pyridin-3-yl)boronic acid 
   (2-fluoro-4-methyl-5-(pyrrolidin-1-ylsulfonyl)phenyl)boronic acid 
   (2-fluoro-4-methyl-5-(morpholinosulfonyl)phenyl)boronic acid 
   N-(2-fluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-2-morpholinoacetamide 
   2-chloro-N-(2-fluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acetamide 
   (2-fluoro-5-((4-methylpiperazin-1-yl)methyl)phenyl)boronic acid 
   (2-fluoro-5-(((4-methoxybenzyl)amino)methyl)phenyl)boronic acid 
   (5-(((2,4-dimethoxybenzyl)amino)methyl)-2-fluorophenyl)boronic acid 
   (4-((4-ethylpiperazin-1-yl)sulfonyl)naphthalen-1-yl)boronic acid 
   (4-(N-cyclopropylsulfamoyl)naphthalen-1-yl)boronic acid 
   (4-((4-methylpiperidin-1-yl)sulfonyl)naphthalen-1-yl)boronic acid 
   (4-(N-cyclohexylsulfamoyl)naphthalen-1-yl)boronic acid 
   (4-((4-(tert-butoxycarbonyl)piperazin-1-yl)sulfonyl)naphthalen-1-yl)boronic acid 
   (4-(N-isopropylsulfamoyl)naphthalen-1-yl)boronic acid 
   tert-butyl 4-(2-oxo-2-((4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)amino)ethyl)piperazine-1-carboxylate 
   2-(4-methylpiperidin-1-yl)-N-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acetamide 
   (4-(4-(tert-butoxycarbonyl)piperazine-1-carbonyl)-3-chlorophenyl)boronic acid 
   (5-((diethylamino)methyl)-2-fluorophenyl)boronic acid 
   (4-(N,N-dimethylsulfamoyl)naphthalen-1-yl)boronic acid 
   (4-(N-cyclopentylsulfamoyl)naphthalen-1-yl)boronic acid 
   (E)-ethyl 3-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acrylate 
   (E)-3-(3-boronophenyl)acrylic acid 
   (E)-ethyl 3-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acrylate 
   potassium trifluoro(3-((4-methoxyphenyl)amino)-3-oxopropyl)borate 
   (3-(1-(4-(2-((tert-butyldimethylsilyl)oxy)ethyl)piperazin-1-yl)ethyl)phenyl)boronic acid 
   2-(dimethylamino)-N-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acetamide 
   2-(diethylamino)-N-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acetamide 
   2-(pyrrolidin-1-yl)-N-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acetamide 
   4-methyl-1-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 
   2-morpholino-N-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acetamide 
   2-chloro-N-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)acetamide 
   (3-(4-(tert-butoxycarbonyl)piperazine-1-carbonyl)-4-fluorophenyl)boronic acid 
   (5-(ethoxymethyl)-2-fluorophenyl)boronic acid 
   (2-fluoro-5-(morpholinomethyl)phenyl)boronic acid 
   (3-(N-(2,4-dimethoxybenzyl)sulfamoyl)phenyl)boronic acid 
   (6-bromo-1-(tert-butoxycarbonyl)-1H-indol-2-yl)boronic acid 
   (3-(N-cyclohexylsulfamoyl)phenyl)boronic acid 
   2-fluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 
   (3-(N-benzylsulfamoyl)phenyl)boronic acid 
   potassium (3-chloro-2-(4-methylpiperidin-1-yl)pyridin-4-yl)trifluoroborate 
   potassium (2-(4-(tert-butoxycarbonyl)piperazin-1-yl)-3-chloropyridin-4-yl)trifluoroborate 
   (3-chloro-4-(4-hydroxypiperidine-1-carbonyl)phenyl)boronic acid 
   (4-fluoro-3-(4-oxopiperidine-1-carbonyl)phenyl)boronic acid 
   (3-fluoro-5-((4-methoxybenzyl)carbamoyl)phenyl)boronic acid 
   (3-(tert-butylcarbamoyl)-5-fluorophenyl)boronic acid 
   (4-chloro-3-(cyclopentylcarbamoyl)phenyl)boronic acid 
   (3-fluoro-5-(isopropylcarbamoyl)phenyl)boronic acid 
   (3-((2-(dimethylamino)ethyl)carbamoyl)-5-fluorophenyl)boronic acid 
   (3-fluoro-5-(4-methylpiperazine-1-carbonyl)phenyl)boronic acid 
   (3-(4-(tert-butoxycarbonyl)piperazine-1-carbonyl)-4-chlorophenyl)boronic acid 
   (4-(morpholinosulfonyl)naphthalen-1-yl)boronic acid 
   (4-(difluoromethoxy)phenyl)boronic acid 
   (3-fluoro-4-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)boronic acid hydrochloride 
   1-cyclopropyl-3-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)urea 
   tert-butyl4-((3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)carbamoyl)piperazine-1-carboxylate 
   (4-(N-cyclopentylsulfamoyl)-3-fluorophenyl)boronic acid 
   (3-fluoro-4-((4-methylpiperidin-1-yl)sulfonyl)phenyl)boronic acid 
   (4-(3-(4-(tert-butoxycarbonyl)piperazin-1-yl)propoxy)-3-fluorophenyl)boronic acid 
   1,1-diethyl-3-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)urea 
   1,1-dimethyl-3-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)urea 
   4-methyl-N-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine-1-carboxamide 
   (4-(1H-pyrrole-1-carboxamido)phenyl)boronic acid 
   (4-((4-(2-hydroxyethyl)piperazin-1-yl)sulfonyl)-3,5-dimethylphenyl)boronic acid 
   (3-((4-ethylpiperazin-1-yl)sulfonyl)-4-methylphenyl)boronic acid 
   6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-benzo[d]imidazole hydrochloride 
   (2,4-dibutoxyphenyl)boronic acid 
   (2-iodophenyl)boronic acid 
   4-hydroxy-N-(3-(4,4,5-trimethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine-1-carboxamide 
   4-methyl-N-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine-1-carboxamide 
   (3-chloro-4-(4-methylpiperidine-1-carbonyl)phenyl)boronic acid 
   (3-(cyclopentylcarbamoyl)-4-fluorophenyl)boronic acid 
   (3-(cyclopropylcarbamoyl)-4-fluorophenyl)boronic acid 
   (3-(((2,4-dimethoxybenzyl)amino)methyl)-5-fluorophenyl)boronic acid 
   (4-(N-(2,4-dimethoxybenzyl)sulfamoyl)phenyl)boronic acid 
   6-butyl-2-(2,4-difluorophenyl)-1,3,6,2-dioxazaborocane 
   6-butyl-2-(3,5-difluorophenyl)-1,3,6,2-dioxazaborocane 
   (4-(N-cyclopentylsulfamoyl)-3,5-dimethylphenyl)boronic acid 
   (4-(2-((tert-butoxycarbonyl)(cyclohexyl)amino)ethoxy)-3-fluorophenyl)boronic acid 
   (3-fluoro-4-(2-(isopropylamino)ethoxy)phenyl)boronic acid 
   (2-fluoro-4-((4-methylpiperazin-1-yl)methyl)phenyl)boronic acid 
   (4-(2-(cyclohexylamino)ethoxy)-3-fluorophenyl)boronic acid 
   (4-(N-(tert-butyl)sulfamoyl)-2-fluorophenyl)boronic acid 
   (2-(2-(dimethylamino)ethoxy)phenyl)boronic acid 
   (4-(N-cyclopropylsulfamoyl)-2-fluorophenyl)boronic acid 
   (3-(N-(tert-butyl)sulfamoyl)-4-methylphenyl)boronic acid 
   (2-fluoro-5-((4-methylpiperidin-1-yl)sulfonyl)phenyl)boronic acid 
   (4-(((tert-butoxycarbonyl)(cyclohexyl)amino)methyl)-2-fluorophenyl)boronic acid 
   3-(benzylcarbamoyl)phenylboronic acid 
   (3-fluoro-4-(morpholinosulfonyl)phenyl)boronic acid 
   1-methyl-3-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)urea 
   4-fluoro -3-(4-methylpiperazine-1-carbonyl)- phenyl boronic acid 
   (4-((4-(2-((tert-butyldiphenylsilyl)oxy)ethyl)piperazin-1-yl)methyl)-2-fluorophenyl)boronic acid 
   (2-fluoro-5-((4-hydroxypiperidin-1-yl)sulfonyl)phenyl)boronic acid 
   (3-chloro-4-(3-(cyclopropylamino)propoxy)phenyl)boronic acid 
   (4-((4-((tert-butyldiphenylsilyl)oxy)piperidin-1-yl)methyl)-2-fluorophenyl)boronic acid 
   (4-(1-(4-hydroxypiperidin-1-yl)ethyl)phenyl)boronic acid 
   (4-(1-(4-((tert-butyldiphenylsilyl)oxy)piperidin-1-yl)ethyl)phenyl)boronic acid 
   (4-(3-((tert-butoxycarbonyl)(cyclopropyl)amino)propoxy)-3-chlorophenyl)boronic acid 
   (2-fluoro-4-((4-hydroxypiperidin-1-yl)methyl)phenyl)boronic acid 
   (4-(((tert-butoxycarbonyl)(cyclopentyl)amino)methyl)-2-fluorophenyl)boronic acid 
   (4-(1-((tert-butoxycarbonyl)(4-methoxybenzyl)amino)ethyl)phenyl)boronic acid 
   (4-((4-(tert-butoxycarbonyl)piperazin-1-yl)methyl)-2-fluorophenyl)boronic acid 
   (4-(N-cyclopropylsulfamoyl)-3-fluorophenyl)boronic acid 
   (4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)-3-fluorophenyl)boronic acid 
   (3-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)-4-methoxyphenyl)boronic acid 
   (4-fluoro-3-(4-hydroxypiperidine-1-carbonyl)phenyl)boronic acid 
   (5-(N-(tert-butyl)sulfamoyl)-2-methoxyphenyl)boronic acid 
   (4-(N,N-dimethylsulfamoyl)-3-fluorophenyl)boronic acid 
   (3-fluoro-4-(N-isopropylsulfamoyl)phenyl)boronic acid 
   (3-(1-(4-(tert-butoxycarbonyl)piperazin-1-yl)ethyl)phenyl)boronic acid 
   (4-fluoro-3-(isopropoxymethyl)phenyl)boronic acid 
   (4-((4-((tert-butyldimethylsilyl)oxy)piperidin-1-yl)sulfonyl)-2-fluorophenyl)boronic acid 
   (4-((cyclopropylamino)methyl)-3-fluorophenyl)boronic acid hydrochloride 
   (4-(((tert-butoxycarbonyl)(cyclopentyl)amino)methyl)-3-fluorophenyl)boronic acid 
   (3-fluoro-4-morpholinophenyl)boronic acid 
   (4-chloro-3-(4-oxopiperidine-1-carbonyl)phenyl)boronic acid 
   (4-(2-(cyclopentylamino)ethoxy)-3-fluorophenyl)boronic acid 
   (4-(2-((tert-butoxycarbonyl)(cyclopentyl)amino)ethoxy)-3-fluorophenyl)boronic acid 
   (3-fluoro-4-(N-methylsulfamoyl)phenyl)boronic acid 
   (3-fluoro-4-((4-methylpiperazin-1-yl)sulfonyl)phenyl)boronic acid 
   (3-(1-(4-ethylpiperazin-1-yl)ethyl)phenyl)boronic acid 
   (4-(N-(tert-butyl)sulfamoyl)-3-fluorophenyl)boronic acid 
   (2-methyl-5-((4-methylpiperazin-1-yl)sulfonyl)phenyl)boronic acid 
   (4-methoxy-3-(N-methoxysulfamoyl)phenyl)boronic acid 
   (4-chloro-3-(4-(2-hydroxyethyl)piperazine-1-carbonyl)phenyl)boronic acid 
   (4-chloro-3-(4-hydroxypiperidine-1-carbonyl)phenyl)boronic acid 
   (6-bromo-2,3-difluoro-4-methoxyphenyl)boronic acid 
   4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzaldehyde 
   (2-fluoro-5-(methoxymethyl)phenyl)boronic acid 
   (3-(2-(4-ethylpiperazin-1-yl)ethoxy)phenyl)boronic acid 
   (4-bromo-2-fluorophenyl)boronic acid 
   (3-chloro-4-(3-fluoropropoxy)phenyl)boronic acid 
   4,4,5,5-tetramethyl-2-(3-nitrophenyl)-1,3,2-dioxaborolane 
   (3-chloro-4-(2-ethoxyethoxy)phenyl)boronic acid 
   (2-fluoro-4-((4-methylpiperidin-1-yl)methyl)phenyl)boronic acid 
   3-(4-ethylpiperazine-1-carbonyl)-4-fluoro phenyl boronic acid 
   (4-(methoxy(methyl)carbamoyl)phenyl)boronic acid 
   (3-(4-ethylpiperazin-1-yl)-5-fluorophenyl)boronic acid 
   (3-((4-(2-hydroxyethyl)piperazin-1-yl)sulfonyl)-4-methylphenyl)boronic acid 
   (2-methoxy-5-(piperazin-1-ylsulfonyl)phenyl)boronic acid hydrochloride 
   (5-((4-(tert-butoxycarbonyl)piperazin-1-yl)sulfonyl)-2-methoxyphenyl)boronic acid 
   (3-fluoro-5-(4-methylpiperidin-1-yl)phenyl)boronic acid 
   (4-chloro-3-(4-ethylpiperazine-1-carbonyl)phenyl)boronic acid 
   potassium (3-chloro-2-morpholinopyridin-4-yl)trifluoroborate 
   (2-ethoxypyrimidin-5-yl)boronic acid 
   (2-(cyclopropylamino)pyrimidin-5-yl)boronic acid 
   (3-(N-(tert-butyl)sulfamoyl)-4-methoxyphenyl)boronic acid 
   (6-(2-methoxyethoxy)pyridin-3-yl)boronic acid 
   potassium trifluoro(3-fluoro-2-morpholinopyridin-4-yl)borate 
   (3-((1-(tert-butoxycarbonyl)piperidin-4-yl)carbamoyl)phenyl)boronic acid 
   (3-chloro-4-((4-oxopiperidin-1-yl)methyl)phenyl)boronic acid 
   2-Benzyloxy-pyridine-5-boronic acid 
   (4-(((tert-butoxycarbonyl)(cyclopropyl)amino)methyl)-3-fluorophenyl)boronic acid 
   (3-(N-cyclopentylsulfamoyl)-4-methylphenyl)boronic acid 
   (5-(N-cyclopentylsulfamoyl)-2-methoxyphenyl)boronic acid 
   (3-(N-cyclopropylsulfamoyl)-4-methylphenyl)boronic acid 
   (5-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)-2-methoxyphenyl)boronic acid 
   (5-(N,N-diethylsulfamoyl)-2-methoxyphenyl)boronic acid 
   (5-(N,N-dimethylsulfamoyl)-2-methoxyphenyl)boronic acid 
   (4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-3-chlorophenyl)boronic acid 
   3-(cyclopropylcarbamoyl)-5-fluorophenylboronic acid 
   (3-bromo-5-ethoxyphenyl)boronic acid 
   (3-chloro-4-(cyclohexylcarbamoyl)phenyl)boronic acid 
   2-fluoro-3-(morpholine-4-carbonyl)phenylboronic acid 
   (3-(cyclohexylcarbamoyl)-4-fluorophenyl)boronic acid 
   (3-(dimethylcarbamoyl)-4-fluorophenyl)boronic acid 
   (3-fluoro-4-(3-fluoropropoxy)phenyl)boronic acid 
   (4-ethoxy-6-methylpyridin-3-yl)boronic acid 
   (3-(3-fluoropropoxy)-4-methylphenyl)boronic acid 
   3,3-difluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)indolin-2-one 
   (4-(2-(4-((tert-butyldiphenylsilyl)oxy)piperidin-1-yl)ethoxy)-3-fluorophenyl)boronic acid 
   (4-(2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethoxy)-3-fluorophenyl)boronic acid 
   (3-fluoro-4-(2-(4-hydroxypiperidin-1-yl)ethoxy)phenyl)boronic acid 
   (3-fluoro-4-(2-(4-oxopiperidin-1-yl)ethoxy)phenyl)boronic acid 
   (4-((4-((tert-butyldiphenylsilyl)oxy)piperidin-1-yl)methyl)phenyl)boronic acid 
   (4-methoxy-3-(N-((4-methoxycyclohexyl)methyl)sulfamoyl)phenyl)boronic acid 
   (4-(2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethoxy)-3-chlorophenyl)boronic acid 
   (4-chloro-3-(4-methylpiperazine-1-carbonyl)phenyl)boronic acid 
   (2-morpholinopyridin-4-yl)boronic acid 
   (3-chloro-4-(piperazin-1-ylmethyl)phenyl)boronic acid hydrochloride 
   (4-((4-(tert-butoxycarbonyl)piperazin-1-yl)methyl)-3-chlorophenyl)boronic acid 
   (4-chloro-3-((4-methylpiperazin-1-yl)methyl)phenyl)boronic acid 
   (4-fluoro-3-morpholinophenyl)boronic acid 
   (4-(1-(4-(2-((tert-butyldiphenylsilyl)oxy)ethyl)piperazin-1-yl)ethyl)phenyl)boronic acid 
   (4-(3-(4-((tert-butyldiphenylsilyl)oxy)piperidin-1-yl)propoxy)-3-chlorophenyl)boronic acid 
   (4-(2-(dimethylamino)ethoxy)-3-fluorophenyl)boronic acid 
   (4-(2-(4-ethylpiperazin-1-yl)ethoxy)-3-fluorophenyl)boronic acid 
   (4-(1-(cyclopropylamino)ethyl)phenyl)boronic acid hydrochloride 
   (4-(1-((tert-butoxycarbonyl)(cyclopropyl)amino)ethyl)phenyl)boronic acid 
   (4-(1-aminoethyl)phenyl)boronic acid hydrochloride 
   (4-methoxy-3-nitrophenyl)boronic acid 
   (3-(tert-butylcarbamoyl)-4-chlorophenyl)boronic acid 
   (2-(3-fluoropropoxy)-4-(trifluoromethoxy)phenyl)boronic acid 
   (4-chloro-3-(isopropylcarbamoyl)phenyl)boronic acid 
   (4-chloro-3-(cyclohexylcarbamoyl)phenyl)boronic acid 
   (3-(cyclohexylcarbamoyl)-5-fluorophenyl)boronic acid 
   4-(4-ethylpiperazine-1-carbonyl)-3-fluorophenylboronic acid 
   (3-fluoro-5-(4-methylpiperazin-1-yl)phenyl)boronic acid 
   (3-(4-((tert-butyldimethylsilyl)oxy)piperidin-1-yl)-5-fluorophenyl)boronic acid 
   (2-(4-methylpiperidin-1-yl)pyrimidin-5-yl)boronic acid 
   (3-(cyclohexylcarbamoyl)phenyl)boronic acid 
   (4-(isopropylcarbamoyl)phenyl)boronic acid 
   (2-(4-ethylpiperazin-1-yl)pyrimidin-5-yl)boronic acid 
   (3-chloro-4-(2-morpholinoethoxy)phenyl)boronic acid 
   (4-fluoro-3-(pyrrolidin-1-yl)phenyl)boronic acid 
   (3-(N-cyclohexylsulfamoyl)-4-methoxyphenyl)boronic acid 
   (3-(N-isopropylsulfamoyl)-4-methoxyphenyl)boronic acid 
   (4-(((1-(tert-butoxycarbonyl)piperidin-4-yl)oxy)methyl)phenyl)boronic acid 
   (3-fluoro-4-(3-(4-methylpiperazin-1-yl)propoxy)phenyl)boronic acid hydrochloride 
   (3-fluoro-4-(3-(4-methylpiperidin-1-yl)propoxy)phenyl)boronic acid hydrochloride 
   (3-fluoro-4-(3-(piperazin-1-yl)propoxy)phenyl)boronic acid hydrochloride 
   1-methyl-3-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)urea 
   (3-amino-4-fluorophenyl)boronic acid hydrochloride 
   (3-((tert-butoxycarbonyl)amino)-4-fluorophenyl)boronic acid 
   (3-(dibenzylamino)-4-fluorophenyl)boronic acid 
   (3-morpholino-5-(trifluoromethyl)phenyl)boronic acid 
   (3-(difluoromethyl)-4-fluorophenyl)boronic acid 
   (2-(3-fluoropropoxy)phenyl)boronic acid 
   2-(5-(difluoromethyl)-2-fluorophenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 
   ethyl (3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)carbamate 
   methyl (3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)carbamate 
   methyl (4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)carbamate 
   4-bromo-2,5-difluorophenylboronic acid 
   3-fluoro-4-(4-oxopiperidine-1-carbonyl)phenylboronic acid 
   4-(4-(tert-butoxycarbonyl)piperazine-1-carbonyl)-3-fluorophenylboronic acid 
   (4-(2-((tert-butoxycarbonyl)(cyclopropyl)amino)ethoxy)-3-fluorophenyl)boronic acid 
   (4-(2-(4-(2-((tert-butyldiphenylsilyl)oxy)ethyl)piperazin-1-yl)ethoxy)-3-fluorophenyl)boronic acid 
   (3-chloro-4-(3-(4-methylpiperidin-1-yl)propoxy)phenyl)boronic acid 
   (4-(2-(diethylamino)ethoxy)-3-fluorophenyl)boronic acid 
   (3-(N-isopropylsulfamoyl)-4-methylphenyl)boronic acid 
   (4-methyl-3-((4-methylpiperazin-1-yl)sulfonyl)phenyl)boronic acid 
   (2-methoxy-5-(methoxysulfonyl)phenyl)boronic acid 
   (3-fluoro-4-(2-(4-methylpiperazin-1-yl)ethoxy)phenyl)boronic acid 
   (3-(N,N-dimethylsulfamoyl)-4-methoxyphenyl)boronic acid 
   (5-(N-cyclohexylsulfamoyl)-2-methoxyphenyl)boronic acid 
   (4-(1-(4-methylpiperazin-1-yl)ethyl)phenyl)boronic acid 
   (4-carbamoyl-3-chlorophenyl)boronic acid 
   (3-fluoro-5-(piperazin-1-ylmethyl)phenyl)boronic acid hydrochloride 
   (3-((3-methoxyphenyl)carbamoyl)phenyl)boronic acid 
   (4-((2-methoxyphenyl)carbamoyl)phenyl)boronic acid 
   (3-((3-(trifluoromethoxy)phenyl)carbamoyl)phenyl)boronic acid 
   (4-(N-cyclohexylsulfamoyl)phenyl)boronic acid 
   (3-chloro-4-(3-(4-ethylpiperazin-1-yl)propoxy)phenyl)boronic acid 
   (3-chloro-4-(3-(4-methylpiperazin-1-yl)propoxy)phenyl)boronic acid 
   (5-((4-((tert-butyldiphenylsilyl)oxy)piperidin-1-yl)sulfonyl)-2-methoxyphenyl)boronic acid 
   (2-methoxy-5-(N-methylsulfamoyl)phenyl)boronic acid 
   (3-fluoro-4-((4-hydroxypiperidin-1-yl)methyl)phenyl)boronic acid 
   (3-((4-(2-((tert-butyldiphenylsilyl)oxy)ethyl)piperazin-1-yl)sulfonyl)-4-methoxyphenyl)boronic acid 
   4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline hydrochloride 
   4,4,5,5-tetramethyl-2-(4-nitrophenyl)-1,3,2-dioxaborolane 
   (2,4-difluoro-3-(methoxycarbonyl)phenyl)boronic acid 
   1-(2-methoxyethyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)indoline 
   (3,5-difluoro-4-(methoxycarbonyl)phenyl)boronic acid 
   1-benzyl-3,3-difluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)indolin-2-one 
   (3-carbamoyl-5-fluorophenyl)boronic acid 
   (3-(dimethylcarbamoyl)-5-fluorophenyl)boronic acid 
   (4-(3-ethoxy-3-oxopropyl)phenyl)boronic acid 
   (E)-(4-(3-ethoxy-3-oxoprop-1-en-1-yl)phenyl)boronic acid 
   3-(3-boronophenyl)propanoic acid 
   (4-((4-methoxybenzyl)carbamoyl)phenyl)boronic acid 
   3-(Cyclopentylcarbamoyl)phenylboronic acid 
   (3-((4-methoxybenzyl)carbamoyl)phenyl)boronic acid 
   (4-(cyclopentylcarbamoyl)phenyl)boronic acid 
   (4-((furan-2-ylmethyl)carbamoyl)phenyl)boronic acid 
   2,2,2-trifluoroacetic acid compound with (4-(1-(piperazin-1-yl)ethyl)phenyl)boronic acid (1:1) 
   (4-(1-(4-(tert-butoxycarbonyl)piperazin-1-yl)ethyl)phenyl)boronic acid 
   (4-(cyclopropylcarbamoyl)phenyl)boronic acid 
   (3-(N-cyclopentylsulfamoyl)-4-methoxyphenyl)boronic acid 
   (3-((4-hydroxypiperidin-1-yl)sulfonyl)-4-methoxyphenyl)boronic acid 
   (3-((4-(tert-butoxycarbonyl)piperazin-1-yl)sulfonyl)-4-methoxyphenyl)boronic acid 
   (3-amino-4-fluorophenyl)boronic acid 
   (3-(N,N-diethylsulfamoyl)-4-methoxyphenyl)boronic acid 
   (4-methoxy-3-((4-methylpiperazin-1-yl)sulfonyl)phenyl)boronic acid 
   (3-chloro-4-(2-(4-hydroxypiperidin-1-yl)ethoxy)phenyl)boronic acid 
   (3-chloro-4-(2-(diethylamino)ethoxy)phenyl)boronic acid 
   (3-fluoro-4-(2-morpholinoethoxy)phenyl)boronic acid 
   (4-((4-methylpiperazin-1-yl)methyl)phenyl)boronic acid 
   (4-methoxy-3-(N-methylsulfamoyl)phenyl)boronic acid 
   (3-((4-ethylpiperazin-1-yl)sulfonyl)-4-methoxyphenyl)boronic acid 
   (5-((4-ethylpiperazin-1-yl)sulfonyl)-2-methoxyphenyl)boronic acid 
   (2-methoxy-5-((4-methylpiperidin-1-yl)sulfonyl)phenyl)boronic acid 
   (4-(3-(dimethylamino)propoxy)-3-fluorophenyl)boronic acid hydrochloride 
   (4-chloro-3-((4-methylpiperidin-1-yl)methyl)phenyl)boronic acid 
   (5-(N-cyclopropylsulfamoyl)-2-methoxyphenyl)boronic acid 
   (2-methoxy-5-((4-methylpiperazin-1-yl)sulfonyl)phenyl)boronic acid 
   (3-chloro-4-(morpholinomethyl)phenyl)boronic acid 
   3-fluoro-4-(4-methylpiperidine-1-carbonyl)phenylboronic acid 
   (4-methyl-6-(pyrrolidin-1-yl)pyridin-3-yl)boronic acid 
   (4-(1-(4-(2-((tert-butyldimethylsilyl)oxy)ethyl)piperazin-1-yl)ethyl)phenyl)boronic acid 
   (3-chloro-4-(2-(dimethylamino)ethoxy)phenyl)boronic acid 
   2-Benzyloxypyrimidine-5-boronic acid 
   (4-Fluoro-3-(methylcarbamoyl)phenyl)boronic acid 
   (4-(1-(4-((tert-butyldimethylsilyl)oxy)piperidin-1-yl)ethyl)phenyl)boronic acid 
   (4-(1-(4-ethylpiperazin-1-yl)ethyl)phenyl)boronic acid hydrochloride 
   (3-(2-((tert-butyldiphenylsilyl)oxy)ethoxy)phenyl)boronic acid 
   (2-(4-methylpiperidin-1-yl)pyridin-3-yl)boronic acid 
   (5-((4-(2-hydroxyethyl)piperazin-1-yl)sulfonyl)-2-methoxyphenyl)boronic acid 
   (2-methoxy-5-(pyrrolidin-1-ylsulfonyl)phenyl)boronic acid 
   (4-(2-((tert-butoxycarbonyl)(cyclopropyl)amino)ethoxy)phenyl)boronic acid 
   4-((4-fluoro-2-(4,4,5,5-tetramethyl-1,3-dioxolan-2-yl)phenyl)sulfonyl)morpholine 
   (2-(dibenzylamino)phenyl)boronic acid 
   (3-((2-methoxyphenyl)carbamoyl)phenyl)boronic acid 
   (4-chloro-3-(dimethylcarbamoyl)phenyl)boronic acid 
   (1H-indol-6-yl)boronic acid 
   6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole 
   (4-(N-benzylsulfamoyl)phenyl)boronic acid 
   (3-((4-(trifluoromethoxy)phenyl)carbamoyl)phenyl)boronic acid 
   (4-((3-(trifluoromethoxy)phenyl)carbamoyl)phenyl)boronic acid 
   (4-methoxy-3-((4-methylpiperidin-1-yl)sulfonyl)phenyl)boronic acid 
   (3-chloro-4-(3-(dimethylamino)propoxy)phenyl)boronic acid 
   (4-(2-(4-((tert-butyldiphenylsilyl)oxy)piperidin-1-yl)ethoxy)-3-chlorophenyl)boronic acid 
   (3-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-5-fluorophenyl)boronic acid 
   (3-fluoro-5-((4-oxopiperidin-1-yl)methyl)phenyl)boronic acid 
   (4-((methylamino)methyl)phenyl)boronic acid 
   (4-(1-(pyrrolidin-1-yl)ethyl)phenyl)boronic acid 
   (4-(1-(diethylamino)ethyl)phenyl)boronic acid 
   (4-(1-(4-methylpiperazin-1-yl)ethyl)phenyl)boronic acid hydrochloride 
   (4-(1-(dimethylamino)ethyl)phenyl)boronic acid hydrochloride 
   3-(3-(4-ethylpiperazin-1-yl)propoxy)-4-methylphenylboronic acid 
   3-(3-(4-(tert-butoxycarbonyl)piperazin-1-yl)propoxy)-4-methylphenylboronic acid 
   (4-chloro-3-((4-ethylpiperazin-1-yl)methyl)phenyl)boronic acid 
   (3-fluoro-4-(3-(pyrrolidin-1-yl)propoxy)phenyl)boronic acid 
   (4-methyl-3-(3-(piperazin-1-yl)propoxy)phenyl)boronic acid 
   (3-carbamoyl-4-fluorophenyl)boronic acid 
   (3-chloro-4-(ethoxycarbonyl)phenyl)boronic acid 
   (4-((4-bromophenyl)carbamoyl)phenyl)boronic acid 
   4-methyl-3-(3-(4-methylpiperazin-1-yl)propoxy)phenylboronic acid 
   (3-(thiazol-2-ylcarbamoyl)phenyl)boronic acid 
   (3-(methoxy(methyl)carbamoyl)phenyl)boronic acid 
   (4-(thiazol-2-ylcarbamoyl)phenyl)boronic acid 
   4-methyl-3-(3-(4-methylpiperidin-1-yl)propoxy)phenylboronic acid 
   (2-((4-(tert-butoxycarbonyl)piperazin-1-yl)methyl)-5-fluorophenyl)boronic acid 
   (4-carbamoyl-2-fluorophenyl)boronic acid 
   (4-(dimethylcarbamoyl)-2-fluorophenyl)boronic acid 
   (2-fluoro-4-(4-methylpiperidine-1-carbonyl)phenyl)boronic acid 
   4-(cyclohexylcarbamoyl)phenylboronic acid 
   4-(benzylcarbamoyl)phenylboronic acid 
   (4-methoxy-3-(pyrrolidin-1-ylsulfonyl)phenyl)boronic acid 
   (4-(3-chloropropoxy)-3-fluorophenyl)boronic acid 
   (4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)-3-fluorophenyl)boronic acid 
   (4-methoxy-3-(morpholinosulfonyl)phenyl)boronic acid 
   (4-chloro-3-((diethylamino)methyl)phenyl)boronic acid 
   (4-chloro-3-(pyrrolidin-1-ylmethyl)phenyl)boronic acid 
   (3-chloro-4-(3-(pyrrolidin-1-yl)propoxy)phenyl)boronic acid 
   (3-chloro-4-(2-(4-ethylpiperazin-1-yl)ethoxy)phenyl)boronic acid 
   (3-chloro-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)boronic acid 
   (3-chloro-4-((4-hydroxypiperidin-1-yl)methyl)phenyl)boronic acid 
   (3-chloro-4-((4-ethylpiperazin-1-yl)methyl)phenyl)boronic acid 
   (3-chloro-4-((diethylamino)methyl)phenyl)boronic acid 
   (((methylazanediyl)bis(methylene))bis(4,1-phenylene))diboronic acid 
   (3-chloro-4-(2-(4-methylpiperazin-1-yl)ethoxy)phenyl)boronic acid 
   (6-(4-hydroxypiperidin-1-yl)pyridin-3-yl)boronic acid 
   (4-(2-(4-(tert-butoxycarbonyl)piperazin-1-yl)ethoxy)-3-chlorophenyl)boronic acid 
   (3-chloro-4-(2-(piperazin-1-yl)ethoxy)phenyl)boronic acid 
   (4-chloro-3-(4-methylpiperidine-1-carbonyl)phenyl)boronic acid 
   (4-chloro-3-(methylcarbamoyl)phenyl)boronic acid 
   (3-fluoro-5-((2,2,2-trifluoroethoxy)methyl)phenyl)boronic acid 
   (4-chloro-3-(ethoxycarbonyl)phenyl)boronic acid 
   (4-chloro-3-(methoxycarbonyl)phenyl)boronic acid 
   (2-((dimethylamino)methyl)-4-fluorophenyl)boronic acid 
   (4-((4-ethylpiperazin-1-yl)methyl)-2-fluorophenyl)boronic acid 
   (4-(methylcarbamoyl)phenyl)boronic acid 
   (3-(4-(tert-butoxycarbonyl)piperazine-1-carbonyl)phenyl)boronic acid 
   (3-(4-methylpiperidine-1-carbonyl)phenyl)boronic acid 
   2-ethoxy-3-methylphenylboronic acid 
   N-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)pyrrolidine-1-carboxamide 
   (3-chloro-4-(morpholine-4-carbonyl)phenyl)boronic acid 
   4-fluoro-3-pyrrolidine-1-carbonyl phenyl boronic acid 
   4-((4-ethylpiperazin-1-yl)methyl)-3-fluorophenylboronic acid 
   2-(benzyloxy)-4-(trifluoromethoxy)phenylboronic acid 
   2-ethoxy-4-(trifluoromethoxy)phenylboronic acid 
   (4-(2-(4-(tert-butoxycarbonyl)piperazin-1-yl)ethoxy)-3-fluorophenyl)boronic acid 
   3-fluoro-5-(methylcarbamoyl)phenylboronic acid 
   3-(ethoxycarbonyl)-5-fluorophenylboronic acid 
   3-(diethylcarbamoyl)-5-fluorophenylboronic acid 
   (4-((4-(tert-butoxycarbonyl)piperazin-1-yl)methyl)-3-fluorophenyl)boronic acid 
   3-fluoro-5-(morpholine-4-carbonyl)phenylboronic acid 
   (3-(ethoxymethyl)-4-fluorophenyl)boronic acid 
   3-((diethylamino)methyl)-4-fluorophenylboronic acid 
   (5-bromo-1-(tert-butoxycarbonyl)-1H-indol-2-yl)boronic acid 
   4-fluoro-3-(morpholinomethyl)phenylboronic acid 
   (3-((4-(tert-butoxycarbonyl)piperazin-1-yl)methyl)-4-fluorophenyl)boronic acid 
   (3-(diethylcarbamoyl)-4-fluorophenyl)boronic acid 
   (3-(3-fluoropropoxy)phenyl)boronic acid 
   (4-(3-fluoropropoxy)phenyl)boronic acid 
   (3-(pyrrolidine-1-carbonyl)phenyl)boronic acid 
   4-fluoro-2-((2,2,2-trifluoroethoxy)methyl)phenylboronic acid 
   (2-(ethoxymethyl)-4-fluorophenyl)boronic acid 
   (4-fluoro-2-((2-methoxyethoxy)methyl)phenyl)boronic acid 
   2-((diethylamino)methyl)-4-fluorophenylboronic acid 
   (4-ethoxy-3-fluorophenyl)boronic acid 
   (3-chloro-4-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)boronic acid 
   4-fluoro-2-(morpholinomethyl)phenylboronic acid 
   (2-((4-(tert-butoxycarbonyl)piperazin-1-yl)methyl)-4-fluorophenyl)boronic acid 
   (4-fluoro-2-((4-methylpiperazin-1-yl)methyl)phenyl)boronic acid 
   4-fluoro-2-((4-methylpiperidin-1-yl)methyl)phenylboronic acid 
   4-fluoro-2-(pyrrolidin-1-ylmethyl)phenylboronic acid 
   2-morpholino-5-(trifluoromethyl)phenylboronic acid 
   (2-(4-ethylpiperazin-1-yl)-5-(trifluoromethyl)phenyl)boronic acid 
   (4-chloro-3-(cyclopropylcarbamoyl)phenyl)boronic acid 
   (4-Chloro-3-(diethylcarbamoyl)phenyl)boronic acid 
   (4-chloro-3-(pyrrolidine-1-carbonyl)phenyl)boronic acid 
   2-(pyrrolidin-1-yl)-5-(trifluoromethyl)phenylboronic acid 
   (4-chloro-3-(morpholine-4-carbonyl)phenyl)boronic acid 
   (2-fluoro-4-(methylcarbamoyl)phenyl)boronic acid 
   (4-(ethoxycarbonyl)-2-fluorophenyl)boronic acid 
   (4-(cyclopropylcarbamoyl)-2-fluorophenyl)boronic acid 
   (2-fluoro-4-(morpholine-4-carbonyl)phenyl)boronic acid 
   (4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)phenyl)boronic acid 
   ((4-((4-oxopiperidin-1-yl)methyl)phenyl)boronic acid 
   (6-(4-((tert-butyldiphenylsilyl)oxy)piperidin-1-yl)pyridin-3-yl)boronic acid 
   3-fluoro-5-(isopropoxymethyl)phenylboronic acid 
   (4-fluoro-3-((2-methoxyethoxy)methyl)phenyl)boronic acid 
   (3-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)phenyl)boronic acid 
   (3-fluoro-4-(pyrrolidin-1-ylmethyl)phenyl)boronic acid 
   3-(ethoxymethyl)-5-fluorophenylboronic acid 
   (6-((tert-butoxycarbonyl)(methyl)amino)pyridin-3-yl)boronic acid 
   (3-(2-(4-methylpiperazin-1-yl)ethoxy)phenyl)boronic acid 
   (4-(((4-bromobenzyl)(methyl)amino)methyl)phenyl)boronic acid 
   (4-((4-(2-((tert-butyldiphenylsilyl)oxy)ethyl)piperazin-1-yl)methyl)-3-fluorophenyl)boronic acid 
   (3-fluoro-4-((4-methylpiperidin-1-yl)methyl)phenyl)boronic acid 
   3-fluoro-5-(methoxymethyl)phenylboronic acid 
   (4-(2-(4-ethylpiperazin-1-yl)ethoxy)phenyl)boronic acid 
   3-((tert-butoxycarbonyl(cyclopropyl)amino)methyl)-5-fluorophenylboronic acid 
   (3-chloro-2-(4-methylpiperidin-1-yl)pyridin-4-yl)boronic acid 
   (E)-(4-(1-(hydroxyimino)ethyl)phenyl)boronic acid 
   (2-(4-methylpiperidin-1-yl)pyridin-4-yl)boronic acid 
   2-(4-ethylpiperazin-1-ylsulfonyl)phenylboronic acid 
   2-(4-(tert-butoxycarbonyl)piperazin-1-ylsulfonyl)phenylboronic acid 
   2-(4-methylpiperazin-1-ylsulfonyl)phenylboronic acid 
   2-(pyrrolidin-1-ylmethyl)phenylboronic acid 
   (3-(N-cyclopropylsulfamoyl)phenyl)boronic acid 
   (4-(2-(tert-butoxy)-2-oxoethyl)phenyl)boronic acid 
   (3-((4-ethylpiperazin-1-yl)sulfonyl)phenyl)boronic acid 
   (3-(piperazin-1-ylsulfonyl)phenyl)boronic acid 
   3-(4-methylpiperazin-1-ylsulfonyl)phenylboronic acid 
   (3-(3-ethoxypropoxy)phenyl)boronic acid 
   (3-(3-morpholinopropoxy)phenyl)boronic acid 
   3-(3-(4-(tert-butoxycarbonyl)piperazin-1-yl)propoxy)phenylboronic acid 
   (3-(3-(4-methylpiperazin-1-yl)propoxy)phenyl)boronic acid 
   (3-(3-(4-methylpiperidin-1-yl)propoxy)phenyl)boronic acid 
   4-(4-(tert-butoxycarbonyl)piperazin-1-ylsulfonyl)phenylboronic acid 
   (4-((4-(2-hydroxyethyl)piperazin-1-yl)methyl)phenyl)boronic acid 
   (3-(3-(dimethylamino)propoxy)phenyl)boronic acid 
   4-((diethylamino)methyl)phenylboronic acid 
   potassium ((tert-butylamino)methyl)trifluoroborate 
   potassium trifluoro((isopropylamino)methyl)borate 
   potassium trifluoro((4-methylpiperazin-1-yl)methyl)borate 
   potassium trifluoro((4-methylpiperidin-1-yl)methyl)borate 
   potassium trifluoro(morpholinomethyl)borate 
   potassium ((cyclopentylamino)methyl)trifluoroborate 
   potassium trifluoro(3-((3-nitrophenyl)amino)-3-oxopropyl)borate 
   potassium trifluoro(3-((4-nitrophenyl)amino)-3-oxopropyl)borate 
   potassium trifluoro(3-oxo-3-((2-(trifluoromethoxy)phenyl)amino)propyl)borate 
   potassium trifluoro(3-((2-methoxyphenyl)amino)-3-oxopropyl)borate 
   potassium trifluoro(3-oxo-3-((2-(trifluoromethyl)phenyl)amino)propyl)borate 
   (4-(pyrrolidin-1-yl)phenyl)boronic acid 
   (4-(isopropoxymethyl)phenyl)boronic acid 
   potassium trifluoro(3-oxo-3-(phenylamino)propyl)borate 
   potassium trifluoro(3-morpholino-3-oxopropyl)borate 
   potassium trifluoro(3-((2-fluorophenyl)amino)-3-oxopropyl)borate 
   potassium trifluoro(3-((3-fluorophenyl)amino)-3-oxopropyl)borate 
   potassium trifluoro(3-((4-fluorophenyl)amino)-3-oxopropyl)borate 
   potassium (3-((2-bromophenyl)amino)-3-oxopropyl)trifluoroborate 
   potassium (3-((3-bromophenyl)amino)-3-oxopropyl)trifluoroborate 
   4,4,5,5-tetramethyl-2-(3,4,5-trifluorophenyl)-1,3,2-dioxaborolane 
   Potassium (3-((2-chlorophenyl)amino)-3-oxopropyl)trifluoroborate 
   potassium (3-((3-chlorophenyl)amino)-3-oxopropyl)trifluoroborate 
   potassium (3-((4-bromophenyl)amino)-3-oxopropyl)trifluoroborate 
   potassium (3-((4-chlorophenyl)amino)-3-oxopropyl)trifluoroborate 
   N-ethyl-N-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzyl)ethanamine 
   2-(3-(methoxymethyl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 
   (5-fluoro-2-(methoxymethyl)phenyl)boronic acid 
   (2-methoxy-6-(trifluoromethyl)pyridin-3-yl)boronic acid 
   1,1-diethyl-3-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)urea 
   N-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)morpholine-4-carboxamide 
   4-(6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-yl)morpholine 
   2-methoxy-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   potassium trifluoro(3-oxo-3-(p-tolylamino)propyl)borate 
   (4-(difluoromethyl)phenyl)boronic acid 
   (6-(pyrrolidin-1-yl)pyridin-3-yl)boronic acid 
   tert-butyl (4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)carbamate 
   (2,5-dibromopyridin-4-yl)boronic acid 
   2-(2,5-dimethyl-1H-pyrrol-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   (3-(cyclopropylamino)-4,5-difluorophenyl)boronic acid 
   (3,5-dimethyl-4-(pyrrolidin-1-ylsulfonyl)phenyl)boronic acid 
   4-(cyclopropylamino)phenylboronic acid 
   (4-fluoro-3-(methoxymethyl)phenyl)boronic acid 
   (3-(2-(dimethylamino)ethoxy)phenyl)boronic acid 
   (3-(difluoromethyl)phenyl)boronic acid 
   (2-(aminomethyl)phenyl)boronic acid 
   (2-(4-(tert-butoxycarbonyl)piperazin-1-yl)pyridin-4-yl)boronic acid 
   (4-(1-(4-methylpiperidin-1-yl)ethyl)phenyl)boronic acid hydrochloride 
   (4-(1-morpholinoethyl)phenyl)boronic acid hydrochloride 
   2-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)propyl)isoindoline-1,3-dione 
   (3-(aminomethyl)phenyl)boronic acid 
   (E)-(3-((hydroxyimino)methyl)phenyl)boronic acid 
   tert-butyl 4-((4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)carbamoyl)piperazine-1-carboxylate 
   1-(tert-butoxycarbonyl)-1H-indol-2-ylboronic acid 
   (3-(N,N-diethylsulfamoyl)-4-(trifluoromethoxy)phenyl)boronic acid 
   (3-(pyrrolidin-1-ylsulfonyl)-4-(trifluoromethoxy)phenyl)boronic acid 
   (2-((4-ethylpiperazin-1-yl)methyl)-5-fluorophenyl)boronic acid 
   (3-((4-ethylpiperazin-1-yl)methyl)phenyl)boronic acid 
   (3-(1-morpholinoethyl)phenyl)boronic acid 
   (4-((4-ethylpiperazin-1-yl)sulfonyl)phenyl)boronic acid 
   (4-((4-methylpiperidin-1-yl)sulfonyl)phenyl)boronic acid 
   (4-(N,N-diethylsulfamoyl)phenyl)boronic acid 
   (4-(pyrrolidin-1-ylsulfonyl)phenyl)boronic acid 
   (3-(N,N-dimethylsulfamoyl)phenyl)boronic acid 
   (2-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)-4,5-difluorophenyl)boronic acid 
   (2-((diethylamino)methyl)phenyl)boronic acid 
   (3-(3-ethoxypropoxy)-4-methylphenyl)boronic acid 
   (3-(2,2,2-trifluoroethoxy)-5-(trifluoromethyl)phenyl)boronic acid 
   (3-(4-(tert-butoxycarbonyl)piperazin-1-yl)-5-(trifluoromethyl)phenyl)boronic acid 
   (5-fluoro-2-((2,2,2-trifluoroethoxy)methyl)phenyl)boronic acid 
   (2-(ethoxymethyl)-5-fluorophenyl)boronic acid 
   (5-fluoro-2-(pyrrolidin-1-ylmethyl)phenyl)boronic acid 
   (5-fluoro-2-((4-methylpiperazin-1-yl)methyl)phenyl)boronic acid 
   (5-fluoro-2-((4-methylpiperidin-1-yl)methyl)phenyl)boronic acid 
   (2-((dimethylamino)methyl)-5-fluorophenyl)boronic acid 
   (5-fluoro-2-(morpholinomethyl)phenyl)boronic acid 
   (3-((4-methylpiperidin-1-yl)methyl)phenyl)boronic acid 
   (3-(isopropoxymethyl)phenyl)boronic acid 
   (3-(ethoxymethyl)phenyl)boronic acid 
   (3,5-dimethyl-4-((4-methylpiperazin-1-yl)sulfonyl)phenyl)boronic acid 
   2-(morpholinosulfonyl)phenylboronic acid 
   4-methoxy-6-methylpyridin-3-ylboronic acid 
   (3-(4-ethylpiperazin-1-yl)-5-(trifluoromethyl)phenyl)boronic acid 
   (3-(pyrrolidin-1-yl)-5-(trifluoromethyl)phenyl)boronic acid 
   3-(morpholinosulfonyl)phenylboronic acid 
   (3-(pyrrolidin-1-ylmethyl)phenyl)boronic acid 
   (4-(ethoxymethyl)-3-fluorophenyl)boronic acid 
   (4-((4-ethylpiperazin-1-yl)sulfonyl)-3,5-dimethylphenyl)boronic acid 
   4-(2-morpholinoethoxy)phenylboronic acid 
   2-(isopropoxymethyl)phenylboronic acid 
   (4-(N,N-dimethylsulfamoyl)-3,5-dimethylphenyl)boronic acid 
   (3-(2-morpholinoethoxy)phenyl)boronic acid 
   2-morpholino-1-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)indolin-1-yl)ethanone 
   2-chloro-1-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)indolin-1-yl)ethanone 
   (3-((2,2,2-trifluoroethoxy)methyl)phenyl)boronic acid 
   (3-(methoxymethyl)phenyl)boronic acid 
   (3-((4-(tert-butoxycarbonyl)piperazin-1-yl)methyl)phenyl)boronic acid 
   6-morpholinopyridin-3-ylboronic acid 
   5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)indoline 
   tert-butyl 5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)indoline-1-carboxylate 
   2-(ethoxymethyl)phenylboronic acid 
   2-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-benzo[d]imidazol-1-yl)ethanol 
   potassium (2-bromophenyl)trifluoroborate 
   4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)phenylboronic acid 
   2-(3-methoxypropoxy)phenylboronic acid 
   2-(2-methoxyethoxy)phenylboronic acid 
   (4-(N,N-diethylsulfamoyl)-3,5-dimethylphenyl)boronic acid 
   (3-(4-(tert-butoxycarbonyl)piperazin-1-yl)-4,5-difluorophenyl)boronic acid 
   (3-(p-tolylcarbamoyl)phenyl)boronic acid 
   6-bromo-2-fluoro-3-methylphenylboronic acid 
   (3,4-difluoro-5-(pyrrolidin-1-yl)phenyl)boronic acid 
   (3-fluoro-5-morpholinophenyl)boronic acid 
   (4-fluoro-3-((4-hydroxypiperidin-1-yl)methyl)phenyl)boronic acid 
   3-fluoro-4-((4-methylpiperazin-1-yl)methyl)phenylboronic acid 
   (2-(pyrrolidin-1-yl)pyrimidin-5-yl)boronic acid 
   (4-(3-((tert-butoxycarbonyl)(cyclopropyl)amino)propoxy)phenyl)boronic acid 
   (4-(3-(pyrrolidin-1-yl)propoxy)phenyl)boronic acid 
   (2,3-difluoro-4-(4-methylpiperidin-1-yl)phenyl)boronic acid 
   (3-((4-methoxyphenyl)carbamoyl)phenyl)boronic acid 
   (3-((3-(trifluoromethyl)phenyl)carbamoyl)phenyl)boronic acid 
   (4-(4-(4-methylpiperazin-1-yl)butoxy)phenyl)boronic acid 
   5-fluoro-2-(isopropoxymethyl)phenylboronic acid 
   4-(morpholinosulfonyl)phenylboronic acid 
   3-(3-methoxypropoxy)phenylboronic acid 
   3-(3-(diethylamino)propoxy)phenylboronic acid 
   (3-((diethylamino)methyl)phenyl)boronic acid 
   6-(4-(tert-butoxycarbonyl)piperazin-1-yl)pyridin-3-ylboronic acid 
   (3,4-difluoro-5-(4-hydroxypiperidin-1-yl)phenyl)boronic acid 
   (3-(phenylcarbamoyl)phenyl)boronic acid 
   (4-((4-methoxyphenyl)carbamoyl)phenyl)boronic acid 
   (4-((4-fluorophenyl)carbamoyl)phenyl)boronic acid 
   (4-(dibenzylamino)phenyl)boronic acid 
   (3-((3-fluorophenyl)carbamoyl)phenyl)boronic acid 
   4-(morpholinomethyl)phenylboronic acid 
   4-(morpholine-4-carbonyl)phenylboronic acid 
   (3-fluoro-5-(pyrrolidin-1-yl)phenyl)boronic acid 
   (3-(dimethylamino)-5-fluorophenyl)boronic acid 
   (2-(2-morpholinoethoxy)phenyl)boronic acid 
   (4-(2-(diethylamino)ethoxy)phenyl)boronic acid 
   (4-(3-(4-ethylpiperazin-1-yl)propoxy)phenyl)boronic acid 
   1-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-benzo[d]imidazole 
   4-(benzyloxy)phenylboronic acid 
   4-methoxy-2-(methoxymethyl)phenylboronic acid 
   (2-morpholinopyrimidin-5-yl)boronic acid 
   (3-((4-hydroxypiperidin-1-yl)sulfonyl)phenyl)boronic acid 
   (3-(difluoromethyl)-4-methoxyphenyl)boronic acid 
   (2-(N,N-dimethylsulfamoyl)-4,5-difluorophenyl)boronic acid 
   (4-((4-(trifluoromethoxy)phenyl)carbamoyl)phenyl)boronic acid 
   (4-((4-((tert-butyldimethylsilyl)oxy)piperidin-1-yl)sulfonyl)phenyl)boronic acid 
   (2-(N,N-diethylsulfamoyl)-4,5-difluorophenyl)boronic acid 
   (4-((3-fluorophenyl)carbamoyl)phenyl)boronic acid 
   (4-((4-(tert-butoxycarbonyl)piperazin-1-yl)sulfonyl)-3,5-dimethylphenyl)boronic acid 
   (4-morpholinophenyl)boronic acid 
   (Z)-(4-((hydroxyimino)methyl)phenyl)boronic acid 
   (3,5-dimethyl-4-((4-methylpiperidin-1-yl)sulfonyl)phenyl)boronic acid 
   2-(benzyloxy)phenylboronic acid 
   (3,4-difluoro-5-methoxyphenyl)boronic acid 
   1-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole 
   (E)-(2-((hydroxyimino)methyl)phenyl)boronic acid 
   (4-(N-methoxysulfamoyl)-3,5-dimethylphenyl)boronic acid 
   (3-fluoro-4-(methoxymethyl)phenyl)boronic acid 
   3-(benzyloxy)phenylboronic acid 
   (2-(dimethylamino)pyrimidin-5-yl)boronic acid 
   (3,4-difluoro-5-(4-methylpiperazin-1-yl)phenyl)boronic acid 
   2-((4-methylpiperazin-1-yl)methyl)phenylboronic acid 
   (3,5-dimethyl-4-(morpholinosulfonyl)phenyl)boronic acid 
   (3-((4-fluorophenyl)carbamoyl)phenyl)boronic acid 
   (2-((diethylamino)methyl)-5-fluorophenyl)boronic acid 
   2-(morpholinomethyl)phenylboronic acid 
   3-fluoro-4-(morpholine-4-carbonyl)phenylboronic acid 
   (3-((2-fluorophenyl)carbamoyl)phenyl)boronic acid 
   (4-((diethylamino)methyl)-3-fluorophenyl)boronic acid 
   (3-fluoro-4-(morpholinomethyl)phenyl)boronic acid 
   (3-(3-(4-ethylpiperazin-1-yl)propoxy)phenyl)boronic acid 
   2,4-Difluorophenylboronic acid 
   (3,5-dimethyl-4-(N-methylsulfamoyl)phenyl)boronic acid 
   (3-((diisopropylamino)methyl)-4-fluorophenyl)boronic acid 
   (3,4-difluoro-5-morpholinophenyl)boronic acid 
   4-methyl-3-(morpholinosulfonyl)phenylboronic acid 
   N-cyclopropyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzamide 
   (4-methylpiperidin-1-yl)(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)methanone 
   tert-butyl 4-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzoyl)piperazine-1-carboxylate 
   pyrrolidin-1-yl(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)methanone 
   (5-fluoro-2-((4-methylpiperazin-1-yl)methyl)phenyl)boronic acid hydrochloride 
   (3-(3-chloropropoxy)-4-methylphenyl)boronic acid 
   N-cyclopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzamide 
   tert-butyl 4-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzoyl)piperazine-1-carboxylate 
   pyrrolidin-1-yl(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)methanone 
   N,N-diethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzamide 
   morpholino(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)methanone 
   (4-fluoro-2-(methoxymethyl)phenyl)boronic acid 
   (4-methyl-3-(3-morpholinopropoxy)phenyl)boronic acid 
   2-((4-methylpiperidin-1-yl)methyl)phenylboronic acid 
   4-((4-(tert-butoxycarbonyl)piperazin-1-yl)methyl)phenylboronic acid 
   2-(pyrrolidin-1-ylsulfonyl)phenylboronic acid 
   2-fluoro-4-(morpholinomethyl)phenylboronic acid hydrochloride 
   (4-((diethylamino)methyl)-2-fluorophenyl)boronic acid 
   potassium (3-bromophenyl)trifluoroborate 
   potassium (6-bromopyridin-3-yl)trifluoroborate 
   potassium (3-bromopropyl)trifluoroborate 
   potassium (6-bromopyridin-2-yl)trifluoroborate 
   Potassium trifluoro(iodomethyl)borate 
   (4-((4-(2-((tert-butyldimethylsilyl)oxy)ethyl)piperazin-1-yl)sulfonyl)phenyl)boronic acid 
   3-fluoro-5-((2,2,2-trifluoroethoxy)methyl)phenylboronic acid 
   3-((diethylamino)methyl)-5-fluorophenylboronic acid 
   3-fluoro-5-(morpholinomethyl)phenylboronic acid 
   (3-(morpholinosulfonyl)-4-(trifluoromethoxy)phenyl)boronic acid 
   3-(4-(tert-butoxycarbonyl)piperazin-1-ylsulfonyl)-4-methylphenylboronic acid 
   4-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-yl)morpholine 
   4-(dimethylcarbamoyl)-3-fluorophenylboronic acid 
   (3-(morpholine-4-carbonyl)phenyl)boronic acid 
   3-fluoro-4-(3-morpholinopropoxy)phenylboronic acid 
   (4-fluoro-3-(pyrrolidin-1-ylmethyl)phenyl)boronic acid 
   2-methoxy-3-methylphenylboronic acid 
   (4-methyl-3-((4-methylpiperidin-1-yl)sulfonyl)phenyl)boronic acid 
   3-ethoxy-4-methylphenylboronic acid 
   3-fluoro-4-(methoxycarbonyl)phenylboronic acid 
   4-(cyclopropylcarbamoyl)-3-fluorophenylboronic acid 
   (4-((diisopropylamino)methyl)phenyl)boronic acid 
   4-fluoro-3-((4-methylpiperidin-1-yl)methyl)phenylboronic acid 
   (3-((4-methylpiperidin-1-yl)sulfonyl)phenyl)boronic acid 
   (2-(methylamino)pyrimidin-5-yl)boronic acid 
   (3-(tert-butoxymethyl)-4-fluorophenyl)boronic acid 
   3-methoxyphenylboronic acid 
   4-methoxyphenylboronic acid 
   (2-(4-methylpiperidin-1-yl)-5-(trifluoromethyl)phenyl)boronic acid 
   (4-((2-fluorophenyl)carbamoyl)phenyl)boronic acid 
   4-(pyrrolidin-1-ylmethyl)phenylboronic acid 
   (3-(N,N-diethylsulfamoyl)phenyl)boronic acid 
   (4-(2-(4-methylpiperidin-1-yl)ethoxy)phenyl)boronic acid 
   (3-(pyrrolidin-1-ylsulfonyl)phenyl)boronic acid 
   3-borono-2-fluorobenzoic acid 
   4-(3-fluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)morpholine 
   4-(methoxymethyl)phenylboronic acid 
   (2,3-difluorophenyl)boronic acid 
   (4-(3-chloropropoxy)phenyl)boronic acid 
   (4,5-difluoro-2-((4-methylpiperidin-1-yl)sulfonyl)phenyl)boronic acid 
   4-((4-methylpiperidin-1-yl)methyl)phenylboronic acid 
   4-((dimethylamino)methyl)phenylboronic acid 
   4-(ethoxymethyl)phenylboronic acid 
   3-fluoro-4-(pyrrolidine-1-carbonyl)phenylboronic acid 
   2-methoxy-4-(trifluoromethoxy)phenylboronic acid 
   4-(diethylcarbamoyl)-3-fluorophenylboronic acid 
   (3-ethoxy-5-(trifluoromethyl)phenyl)boronic acid 
   (3-(2-(4-hydroxypiperidin-1-yl)ethoxy)phenyl)boronic acid 
   (4-((4-ethylpiperazin-1-yl)methyl)phenyl)boronic acid 
   (3-(N,N-diethylsulfamoyl)-4-methylphenyl)boronic acid 
   (3,4-difluoro-5-(4-methylpiperidin-1-yl)phenyl)boronic acid 
   4-((diMethylaMino)Methyl)-3-fluorophenyl boronic acid 
   (3-(N,N-dimethylsulfamoyl)-4-methylphenyl)boronic acid 
   (3-((4-(tert-butoxycarbonyl)piperazin-1-yl)sulfonyl)phenyl)boronic acid 
   3-(benzyloxy)-4-methylphenylboronic acid 
   (4-(3-(dimethylamino)propoxy)phenyl)boronic acid 
   (4-fluoro-3-((2,2,2-trifluoroethoxy)methyl)phenyl)boronic acid 
   (4-methyl-3-(pyrrolidin-1-ylsulfonyl)phenyl)boronic acid 
   (2-(1,3-dioxolan-2-yl)-4-methoxyphenyl)boronic acid 
   (2-(dimethylamino)-5-(trifluoromethyl)phenyl)boronic acid 
   (4,5-difluoro-2-((4-methylpiperazin-1-yl)sulfonyl)phenyl)boronic acid 
   (3-(4-methylpiperidin-1-yl)-5-(trifluoromethyl)phenyl)boronic acid 
   (3-(dimethylamino)-4,5-difluorophenyl)boronic acid 
   (4,5-difluoro-2-(pyrrolidin-1-ylsulfonyl)phenyl)boronic acid 
   (3-(2-(4-(tert-butoxycarbonyl)piperazin-1-yl)ethoxy)phenyl)boronic acid 
   (4,5-difluoro-2-((4-hydroxypiperidin-1-yl)sulfonyl)phenyl)boronic acid 
   (3,4,5-trifluorophenyl)boronic acid 
   1,1'-Nibenzhydryl-3'-hydroxy-[2,3'-biazetidin]-3-one 
   N-methyl ,propyl-Morpholinium tetrafluoroborate  
   N-methyl ,propyl-Morpholinium iodide 
   N-methyl ,propyl-Morpholinium bromide  
   N-methyl ,ethyl-Morpholinium bis((trifluoromethyl)sulfonyl)imide 
   N-methyl ,ethyl-Morpholinium hexafluorophosphate  
   N-methyl ,ethyl-Morpholinium tetrafluoroborate  
   N-methyl ,ethyl-Morpholinium iodide  
   N-methyl ,ethyl-Morpholinium bromide  
   N-ethyl,methylpyrrolidinium bis((trifluoromethyl)sulfonyl)imide  
   N-ethyl,methylpyrrolidinium trifluoromethanesulfonate  
   N-ethyl,methylpyrrolidinium hexafluorophosphate  
   N-ethyl,methylpyrrolidinium tetrafluoroborate  
   N-ethyl,methylpyrrolidinium bromide  
   N-propyl,methylpyrrolidinium bis((trifluoromethyl)sulfonyl)imide  
   N-propyl,methylpyrrolidinium tetrafluoroborate  
   N-propyl,methylpyrrolidinium hexafluorophosphate  
   N-propyl,methylpyrrolidinium bromide  
   N-butyl,methylpyrrolidinium bis((trifluoromethyl)sulfonyl)imide  
   N-butyl,methylpyrrolidinium perchlorade  
   4-fluoro-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzoic acid 
   6-FLUORO-2-(METHYLSULFANYL)PHENYLBORONIC ACID PINACOL ESTER 
   2-(DIMETHYLAMINO)-5-(4,4,5,5-TETRAMETHYL-1,3,2-DIOXABOROLAN-2-YL)-BENZALDEHYDE 
   3-BORONO-2-METHOXYBENZOIC ACID 
   methyl 4-(trifluoromethyl)-2-methylbenzoate 
   1-(2-fluoro-5-methylpyridin-3-yl)ethanone 
   1-(2-fluoro-5-methylpyridin-3-yl)ethanol 
   2,6-Dimethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 
   (3-(Ethoxycarbonyl)-2-fluorophenyl)boronic acid 
   2-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-4-(trifluoromethyl)aniline 
   (6-chloro-5-methylpyridin-3-yl)boronic acid 
   4-BROMO-2-IODOBENZONITRILE 
   4,4,5,5-tetramethyl-2-(3-(methylthio)-5-(trifluoromethyl)phenyl)-1,3,2-dioxaborolane 
   3,5-Bis(methylthio)pyridine 
   1-bromo-3-chloro-2-iodobenzene 
   5-Bromo-2-methoxy-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 
   2-(3-Isopropylphenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 
   6-Bromo-8-fluoroquinoline 
   1H-indazole-5-boronic acid pinacol ester 
   2-Iodo-5-trifluoromethylpyridine 
   3-Bromo-5-cyclopropylpyridine 
   4-bromo-1-phenyl-1H-pyrazole 
   1-Iodo-3,5-dimethylbenzene 
   2,3,4-Trifluorobromobenzene 
   (4-bromophenyl)trimethylsilane 
   2-Bromo-4-iodoaniline 
   1-bromo-2,4-difluorobenzene 
   5-bromopyridin-2(1H)-one 
   4-bromo-2-iodo-1-methylbenzene 
   5-hexylthiophen-2-boronic acid pinacol ester 
   1,4-dibromo-2-methoxybenzene 
   3-bromo-6-chloro-2-fluorophenol 
   3-fluoro-5-methylphenylboronic acid 
   2,6-dibromobenzaldehyde 
   2-(Benzyloxy)-5-bromo-1,3-dichlorobenzene 
   2-bromo-5-iodophenylboronic acid 
   5-bromo-2-methoxypyridin-3-yl-3-boronic acid 
   4-bromo-2,6-difluorophenol 
   2,3-dimethoxyphenylboronic acid 
   6-bromo-2,3-difluorophenylboronic acid 
   5-bromo-2-fluoropyridin-3-yl-3-boronic acid 
   5-bromo-2-fluoro-3-methylbenzaldehyde 
   5-bromo-1H-pyrazolo[3,4-b]pyridine 
   2,6-dichloropyridine-3-carboxamide 
   1,5-dibromo-2,4-difluorobenzene 
   1-bromo-3-chloro-2-methylbenzene 
   5-Brom-2-methoxy-thioanisol 
   (5-bromo-2-methylphenyl)methanol 
   5-bromo-2-methylbenzaldehyde 
   3,3-difluorocyclobutane-1-carbaldehyde 
   3-iodo-2H-pyrazolo[3,4-b]pyridine 
   5-bromo-2,4-dimethylbenzoic acid 
   METHYL 4-AMINO-5-BROMO-2-METHYLBENZOATE 
   3-bromo-2-fluoro-6-methoxybenzaldehyde 
   2-(1-methylcyclopropyl)ethanol 
   4-fluoro-2-methyl-5-nitroaniline 
   6-(4,4-dimethyl-4,5-dihydro-1,3-oxazol-2-yl)pyridin-2-amine 
   methyl 3-bromo-5-iodobenzoate 
   2-oxaspiro[3.3]heptane-6-carboxylic acid 
   cyclopentanecarbothioamide 
   CYCLOBUTANECARBOTHIOAMIDE 
   cyclopropanecarbothioamide 
   cyclopropanecarboxamide 
   cyclopentanecarboxamide 
   Cyclobutanecarboxamide 
   2-oxaspiro[3.3]heptan-6-amine,hydrochloride 
   (1R,4R)-METHYL 4-FORMYLCYCLOHEXANECARBOXYLATE 
   3,3-dimethylbutan-1-amine hydrochloride 
   4-bromobicyclo[2.2.2]octan-1-amine 
   4-bromobicyclo[2.2.2]octan-1-ol 
   4-bromobicyclo[2.2.2]octane-1-carboxylic acid 
   4-aminobicyclo[2.2.2]octane-1-carbonitrile 
   4-bromobicyclo[2.2.2]octane-1-carbonitrile 
   4-hydroxybicyclo[2.2.2]octane-1-carbonitrile 
   3-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)Benzenamine 
   1-Benzofuran-3-carbonitrile 
   4-AMino-2-broMophenetole 
   2-Bromo-1-ethoxy-4-nitrobenzene 
   8-BROMO-6-CHLORO-9H-PURINE 
   8-BENZYL-3,8-DIAZABICYCLO[3.2.1]OCTANE 
   (1R,2R,4S)-REL-2-AMINO-7-BOC-7-AZABICYCLO[2.2.1]HEPTANE 
   1-METHYLBIGUANIDE SULPHATE 
   5-BROMO-4-CHLOROTHIENO[2,3-D]PYRIMIDINE 
   1-octyl-2,3-dimethylimidazolium hexafluorophosphate  
   1-octyl-2,3-dimethylimidazolium tetrafluoroborate  
   1-octyl-2,3-dimethylimidazolium chloride  
   1-octyl-2,3-dimethylimidazolium bromide  
   N-hexyl-3-metylpyridinium bromide  
   N-hexyl-3-metylpyridinium chloride  
   N-butyl-3-metylpyridinium bis((trifluoromethyl)sulfonyl)imide  
   N-butyl-3-metylpyridinium hexafluorophosphate  
   N-butyl-3-metylpyridinium tetrafluoroborate  
   N-butyl,methylpyrrolidinium trifluoroacetate  
   N-butyl,methylpyrrolidinium hexafluorophosphate  
   N-butyl,methylpyrrolidinium tetrafluoroborate  
   N-butyl,methylpyrrolidinium bromide  
   1-(2’-hydroxylethyl)-3-methylimidazolium tetrafluoroborate  
   1-benzyl-3-methylimidazolium hexafluorophosphate  
   1-benzyl-3-methylimidazolium tetrafluoroborate  
   1-carboxymethyl-3-methylimidazolium chloride  
   1-carboxymethyl-3-methylimidazolium bis(trifluoromethylsulfonyl)imide  
   1-Ethyl ester methyl-3-methylimidazolium bis(trifluoromethylsulfonyl)imide  
   1-Ethyl ester methyl-3-methylimidazolium hexafluorophosphate  
   1-Ethyl ester methyl-3-methylimidazolium tetrafluoroborate  
   1-Ethyl ester methyl-3-methylimidazolium chloride  
   1,3-di(9-chloromethyl anthracene)-3-methylimidazolium chloride  
   1-(9-chloromethyl anthracene)-3-methylimidazolium chloride  
   Amiselimod, MT-1303 
   1H-Benz[e]indolium, 3-[(4-carboxyphenyl)methyl]-1,1,2-trimethyl-, bromide (1:1)  
   Nintedanib Ethanesulfonate Salt 
   Olaparib 
   ONO-4059 analogue 
   ZM241385 
   CP21R7(CP21)  
   SB216763 
   ONO-4059 
   KR-33494 
   3-AZABICYCLO[3.2.1]OCTAN-8-OL HYDROCHLORIDE 
   2-(3-(TERT-BUTOXYCARBONYL)-3-AZABICYCLO[3.2.1]OCTAN-8-YL)ACETIC ACID 
   2-[(TERT-BUTOXY)CARBONYL]-2-AZABICYCLO[2.2.1]HEPTANE-5-CARBOXYLIC ACID 
   TERT-BUTYL 5-OXO-2-AZABICYCLO[2.2.1]HEPTANE-2-CARBOXYLATE 
   EXO-6-HYDROXY-2-AZA-BICYCLO[2.2.1]HEPTANE-2-CARBOXYLIC ACID TERT-BUTYL ESTER 
   (1R,4R,5R)-REL-TERT-BUTYL 5-HYDROXY-2-AZABICYCLO[2.2.1]HEPTANE-2-CARBOXYLATE 
   DIMETHYL 1,4-CUBANEDICARBOXYLATE 
   3-([(TERT-BUTOXY)CARBONYL]AMINO)BICYCLO[1.1.1]PENTANE-1-CARBOXYLIC ACID 
   DIMETHYL BICYCLO[1.1.1]PENTANE-1,3-DICARBOXYLATE 
   3-(METHOXYCARBONYL)BICYCLO[1.1.1]PENTANE-1-CARBOXYLIC ACID 
   Benzofuran-3-carbaldehyde 
   Benzofuran-6-carboxylic acid 
   4-Bromo-5-fluoro-2-methylbenzaldehyde 
   Amiselimod, MT-1303 
   2-(2-Bromoethyl)-1,3-dioxolane 
   Picolinimidamide 
   3-Bromo-2-methylbenzonitrile 
   Tert-butyl 5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate 
   3-Bromo-2-(bromomethyl)pyridine 
   2-Bromo-5-fluoroisonicotinaldehyde 
   2-CHLORO-4-CYANOPHENYLBORONIC ACID PINACOL ESTER 
   BENZYL (4-(HYDROXYMETHYL)BICYCLO[2.2.2]OCTAN-1-YL)CARBAMATE 
   methyl 3-formyl-2-methoxybenzoate 
   (1R)-trans-4-[N-Boc-1-aminoethyl]cyclohexanecarboxylic Acid 
   2-(9H-carbazol-9-yl)acetic acid 
   5-bromo-2,3,3-trimethyl-3H-pyrrolo[2,3-b]pyridine 
   Methyl 4-cyanobicyclo[2.2.2]octane-1-carboxylate 
   N5-((R)-1-((carboxymethyl)amino)-3-(((E)-1,2-dichlorovinyl)thio)-1-oxopropan-2-yl)-L-glutamine 
   4-(Bromomethyl)oxazole hydrobromide 
   4-aminobicyclo[2.2.2]octane-1-carboxylic acid hydrochloride 
   4-DIBENZOTHIOPHENEBORONIC ACID 
   1-chloro-3-phenoxypropan-2-ol 
   (S)-(-)-3-CYCLOHEXENECARBOXYLIC ACID 
   5,7-Dichloropyrido[4,3-d]pyrimidin-4(3H)-one 
   3-methoxypicolinic acid 
   2,4,6-TRIMETHOXY-1,3,5-TRIAZINE 
   Methyl 3-amino-5,6-dimethoxybenzo[b]thiophene-2-carboxylate 
   3,4'-difluoro-[1,1'-biphenyl]-4-amine 
   6-(6-(trifluoromethyl)pyridin-2-yl)-1,3,5-triazine-2,4(1H,3H)-dione 
   N-(3-(2,4-dichlorophenoxy)propyl)-N-methylprop-2-yn-1-amine hydrochloride 
   Tert-butyl 6-fluoro-1H-pyrazolo[3,4-b]pyridine-3-carboxylate  
   4-Methyl-3-nitro-1H-pyrazole 
   2,4,5-Trifluorobenzamidine?hydrochloride 
   2-formyl-1H-indole-6-carbonitrile 
   4-ethyl-2-fluoroaniline 
   1H-Pyrazole, 4-hexyl- 
   tert-butyl (2-(2-(2-bromoethoxy)ethoxy)ethyl)carbamate  
   ethyl 6-cyano-1H-indole-2-carboxylate 
   1-BENZHYDRYLAZETIDIN-3-ONE 
   methyl 2-(2-oxo-1,2,3,4-tetrahydroquinolin-3-yl)acetate 
   4-AMinobicyclo[2.2.2]octan-1-ol hydrochloride 
   3,4-Dimethylbenzonitrile  
   4-aminobicyclo[2.2.2]octane-1-carboxylic acid(盐酸盐形式的有) 
   4-hydroxybicyclo[2.2.2]octane-1-carboxylic acid 
   Acetoacetamide 
   1-Phenyl-3-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole 
   1-Phenyl-1H-pyrazol-3(2H)-one 
   pyrrolidine-2,5-dithione 
   5-Bromo-6-chloro-1H-indole-2-carboxylic acid 
   (1-Methyl-2-oxo-1,2-dihydropyridin-4-yl)boronic acid 
   (2-Amino-4-cyanophenyl)boronic acid hydrochloride 
   (1R,4r)-4-((R)-1-aminoethyl)-N-(pyridin-4-yl)cyclohexane-1-carboxamide dihydrochloride 
   (1R,4r)-4-((R)-1-aminoethyl)-N-(pyridin-4-yl)cyclohexane-1-carboxamide dihydrochloride 
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